Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50139824(7-Chloro-6-hydroxy-pyrido[1,2-a]quinolinylium; chl...)
Affinity DataEC50: >2.00E+5nMAssay Description:Half-Maximal effective concentration of compound required to stimulate of G551D-CFTR activity in the presence of 10 microM FskMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50139824(7-Chloro-6-hydroxy-pyrido[1,2-a]quinolinylium; chl...)
Affinity DataEC50:  1.46E+5nMAssay Description:Half-Maximal effective concentration of compound required to stimulate of wild type-CFTR activity in the presence of 10 microM FskMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed