Affinity DataKi: <0.100nMAssay Description:Inhibition of human cathepsin G using Suc-AAPF-MCA as substrate at pH 7.2 and 298 K measured every 60 secs for 600 secsMore data for this Ligand-Target Pair
Affinity DataKi: 0.150nMAssay Description:Inhibition of cathepsin G (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.174nMAssay Description:Binding affinity against cathepsin GMore data for this Ligand-Target Pair
Affinity DataKi: 0.187nMAssay Description:Binding affinity against cathepsin GMore data for this Ligand-Target Pair
Affinity DataKi: 0.260nMAssay Description:Inhibition of human cathepsin G using Suc-AAPF-MCA as substrate at pH 7.2 and 298 K measured every 60 secs for 600 secsMore data for this Ligand-Target Pair
Affinity DataKi: 0.848nMAssay Description:Binding affinity against cathepsin GMore data for this Ligand-Target Pair
Affinity DataKi: 0.890nMAssay Description:Inhibition of human cathepsin G using Suc-AAPF-MCA as substrate after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 0.916nMAssay Description:Binding affinity against cathepsin GMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Inhibition of human cathepsin G using Suc-AAPF-MCA as substrate after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Inhibition of human cathepsin G using Suc-AAPF-MCA as substrate after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Inhibition of human cathepsin G using Suc-AAPF-MCA as substrate after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 2.90nMAssay Description:Inhibition of human cathepsin G using Suc-AAPF-MCA as substrate after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 3.40nMAssay Description:Inhibition of human cathepsin G using Suc-AAPF-MCA as substrate after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 3.74nMAssay Description:Binding affinity against cathepsin GMore data for this Ligand-Target Pair
Affinity DataKi: 3.85nMAssay Description:Binding affinity against cathepsin GMore data for this Ligand-Target Pair
Affinity DataKi: 3.90nMAssay Description:Binding affinity against cathepsin GMore data for this Ligand-Target Pair
Affinity DataKi: 4.80nMAssay Description:Inhibition of human cathepsin G using Suc-AAPF-MCA as substrate after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 4.90nMAssay Description:Inhibition of human cathepsin G using Suc-AAPF-MCA as substrate after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 7.30nMAssay Description:Inhibition of human cathepsin G using Suc-AAPF-MCA as substrate after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 7.40nMAssay Description:Inhibition of human cathepsin G using Suc-AAPF-MCA as substrate at pH 7.2 and 298 K measured every 60 secs for 600 secsMore data for this Ligand-Target Pair
Affinity DataKi: 8.20nMAssay Description:Inhibition of human cathepsin G using Suc-AAPF-MCA as substrate at pH 7.2 and 298 K measured every 60 secs for 600 secsMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Inhibition of human cathepsin G using Suc-AAPF-MCA as substrate after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Inhibition of human cathepsin G using Suc-AAPF-MCA as substrate after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 14nMAssay Description:Inhibition of human cathepsin G using Suc-AAPF-MCA as substrate at pH 7.2 and 298 K measured every 60 secs for 600 secsMore data for this Ligand-Target Pair
Affinity DataKi: 14.3nMAssay Description:Binding affinity against cathepsin GMore data for this Ligand-Target Pair
Affinity DataKi: 25.3nMAssay Description:Binding affinity against cathepsin GMore data for this Ligand-Target Pair
Affinity DataKi: 38nMAssay Description:Inhibition of human neutrophil Cat GMore data for this Ligand-Target Pair
Affinity DataKi: 38nMAssay Description:Inhibition of cathepsin G in human neutrophils using Suc-Ala-Ala-Pro-Phe-(p-nitroanilide) as substrate for 15 mins by spectrophotometric methodMore data for this Ligand-Target Pair
Affinity DataKi: 44.1nMAssay Description:Binding affinity against cathepsin GMore data for this Ligand-Target Pair
Affinity DataKi: 54nMAssay Description:Inhibition of human cathepsin G using Suc-AAPF-MCA as substrate at pH 7.2 and 298 K measured every 60 secs for 600 secsMore data for this Ligand-Target Pair
Affinity DataKi: 62nMAssay Description:Inhibition of human cathepsin G using Suc-AAPF-MCA as substrate after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 100nM ΔG°: -41.6kJ/molepH: 7.2 T: 2°CAssay Description:Materials: Cathepsin G, 100 mU (VWR, Calbiochem, cat. no. 219373), Substrate Cathepsin G substrate (VWR, Calbiochem, cat. no. 219407). Cathepsin acti...More data for this Ligand-Target Pair
Affinity DataKi: 150nMAssay Description:Inhibition of human cathepsin G using Suc-AAPF-MCA as substrate at pH 7.2 and 298 K measured every 60 secs for 600 secsMore data for this Ligand-Target Pair
Affinity DataKi: 160nMAssay Description:Inhibition of human cathepsin G using Suc-AAPF-MCA as substrate at pH 7.2 and 298 K measured every 60 secs for 600 secsMore data for this Ligand-Target Pair
Affinity DataKi: 160nMAssay Description:Inhibition of human cathepsin G using Suc-AAPF-MCA as substrate after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 200nM ΔG°: -39.8kJ/molepH: 7.2 T: 2°CAssay Description:Materials: Cathepsin G, 100 mU (VWR, Calbiochem, cat. no. 219373), Substrate Cathepsin G substrate (VWR, Calbiochem, cat. no. 219407). Cathepsin acti...More data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:Binding affinity against rat Cathepsin GMore data for this Ligand-Target Pair
Affinity DataKi: 200nMAssay Description:Binding affinity against rat Cathepsin GMore data for this Ligand-Target Pair
Affinity DataKi: 250nMAssay Description:Binding affinity of the compound for human leukocyte cathepsin GMore data for this Ligand-Target Pair
Affinity DataKi: 379nMAssay Description:Inhibitory activity against human cathepsin GMore data for this Ligand-Target Pair
Affinity DataKi: 390nMAssay Description:Inhibition of human cathepsin G using Suc-AAPF-MCA as substrate after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 400nM ΔG°: -38.0kJ/molepH: 7.2 T: 2°CAssay Description:Materials: Cathepsin G, 100 mU (VWR, Calbiochem, cat. no. 219373), Substrate Cathepsin G substrate (VWR, Calbiochem, cat. no. 219407). Cathepsin acti...More data for this Ligand-Target Pair
Affinity DataKi: 410nMAssay Description:Inhibition of human cathepsin G using Suc-AAPF-MCA as substrate after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 480nMAssay Description:Inhibition of human cathepsin G using Suc-AAPF-MCA as substrate after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 490nMAssay Description:Inhibition of human cathepsin G using Suc-AAPF-MCA as substrate after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 500nM ΔG°: -37.4kJ/molepH: 7.2 T: 2°CAssay Description:Materials: Cathepsin G, 100 mU (VWR, Calbiochem, cat. no. 219373), Substrate Cathepsin G substrate (VWR, Calbiochem, cat. no. 219407). Cathepsin acti...More data for this Ligand-Target Pair
Affinity DataKi: 500nM ΔG°: -37.4kJ/molepH: 7.2 T: 2°CAssay Description:Materials: Cathepsin G, 100 mU (VWR, Calbiochem, cat. no. 219373), Substrate Cathepsin G substrate (VWR, Calbiochem, cat. no. 219407). Cathepsin acti...More data for this Ligand-Target Pair
Affinity DataKi: 530nMAssay Description:Inhibition of human cathepsin G using Suc-AAPF-MCA as substrate after 30 minsMore data for this Ligand-Target Pair
Affinity DataKi: 600nM ΔG°: -36.9kJ/molepH: 7.2 T: 2°CAssay Description:Materials: Cathepsin G, 100 mU (VWR, Calbiochem, cat. no. 219373), Substrate Cathepsin G substrate (VWR, Calbiochem, cat. no. 219407). Cathepsin acti...More data for this Ligand-Target Pair
Affinity DataKi: 630nMAssay Description:Inhibition of human cathepsin G using Suc-AAPF-MCA as substrate after 30 minsMore data for this Ligand-Target Pair