Compile Data Set for Download or QSAR
maximum 50k data
Found 5 of ic50 for monomerid = 3044
TargetProtein kinase C beta type(Rattus norvegicus (rat))
Tumor Biology Center

LigandPNGBDBM3044(3-{7-methoxy-23-methyl-12,14-dioxo-3,13,23-triazah...)
Affinity DataIC50:  16nMAssay Description:The activity of PKC, activated by phosphatidylserine and Ca2+, is measured by its ability to transfer phosphate from [gamma-32P]ATP to lysine-rich hi...More data for this Ligand-Target Pair
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TargetMyosin light chain kinase, smooth muscle(Gallus gallus (chicken))
Tumor Biology Center

LigandPNGBDBM3044(3-{7-methoxy-23-methyl-12,14-dioxo-3,13,23-triazah...)
Affinity DataIC50:  49nMpH: 7.2 T: 2°CAssay Description:The activity of MLCK is measured by its ability to transfer 32P from [gamma-32P]ATP to myosin light-chain.More data for this Ligand-Target Pair
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TargetMyosin light chain kinase, smooth muscle(Homo sapiens (Human))
Tumor Biology Center

LigandPNGBDBM3044(3-{7-methoxy-23-methyl-12,14-dioxo-3,13,23-triazah...)
Affinity DataIC50:  200nMAssay Description:Tested for inhibition of Myosin light chain kinase from chicken gizzardMore data for this Ligand-Target Pair
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TargetcGMP-dependent protein kinase 1(Bos taurus (bovine))
Tumor Biology Center

LigandPNGBDBM3044(3-{7-methoxy-23-methyl-12,14-dioxo-3,13,23-triazah...)
Affinity DataIC50: >3.00E+3nMAssay Description:Tested for inhibition of cGMP-dependent protein kinase from bovine lungMore data for this Ligand-Target Pair
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TargetTyrosine-protein kinase Blk(Mus musculus)
Tumor Biology Center

LigandPNGBDBM3044(3-{7-methoxy-23-methyl-12,14-dioxo-3,13,23-triazah...)
Affinity DataIC50: >1.00E+4nMAssay Description:Tested for inhibition of general tyrosine-specific protein kinase activity from murine B cell lysateMore data for this Ligand-Target Pair
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