Affinity DataKi: 2.00E+3nMAssay Description:Competitive inhibition of human recombinant DAAO by Michaelis-Menten plot analysis in presence of D-serineMore data for this Ligand-Target Pair
Affinity DataKi: 7.00E+3nMAssay Description:Inhibition of human recombinant DAO expressed in Escherichia coli BL21(DE3) by oxygraphic assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.09E+4nMAssay Description:Inhibition of human recombinant N-terminal His-tagged DAO expressed in Escherichia coli BL21(DE3) using D-serine as substrate by Lineweaver-Burk plot...More data for this Ligand-Target Pair
Affinity DataKi: 1.38E+4nMAssay Description:Inhibition of mouse Oat6-mediated [3H]ES uptake in Xenopus oocytes after 1 hrMore data for this Ligand-Target Pair
Affinity DataKi: 2.44E+4nMAssay Description:Inhibition of Candida albicans Nce103More data for this Ligand-Target Pair
Affinity DataKi: 3.00E+4nMAssay Description:Binding affinity against human cytosolic Carbonic anhydrase IIMore data for this Ligand-Target Pair
Affinity DataKi: 3.00E+4nMAssay Description:Inhibition of human carbonic anhydrase2More data for this Ligand-Target Pair
TargetCarbonic anhydrase [110-330](Flaveria bidentis (Coastal plain yellowtops))
Istituto Di Biostrutture E Bioimmagini-Cnr
Istituto Di Biostrutture E Bioimmagini-Cnr
Affinity DataKi: 6.45E+4nM ΔG°: -23.5kJ/molepH: 8.3 T: 2°CAssay Description:Inhibition constants of carboxylate inhibitors against F. bidentis CA I were determined by a stopped flow CO2 hydration assay at 20 °C.More data for this Ligand-Target Pair
Affinity DataKi: 7.47E+4nMAssay Description:Binding affinity against human cytosolic Carbonic anhydrase IVMore data for this Ligand-Target Pair
Affinity DataKi: 2.53E+5nMAssay Description:Inhibition of mouse Oat1-mediated [3H]PAH uptake in Xenopus oocytes after 1 hrMore data for this Ligand-Target Pair
Affinity DataKi: 7.30E+5nMAssay Description:Inhibition of human cytosolic carbonic anhydrase 1 by stopped flow CO2 hydration assayMore data for this Ligand-Target Pair
Affinity DataKi: 7.01E+6nMAssay Description:Binding affinity against human cytosolic Carbonic anhydrase VMore data for this Ligand-Target Pair
Affinity DataKi: >1.50E+8nMAssay Description:Binding affinity against human cytosolic Carbonic anhydrase IXMore data for this Ligand-Target Pair