Affinity DataIC50: 0.00700nMAssay Description:Antagonist activity at human AVPR2 by PathHunter beta-arrestin assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.60nMAssay Description:Antagonist activity at human OXTR expressed in CHO-K1 cells by PathHunter beta-arrestin assayMore data for this Ligand-Target Pair
Affinity DataIC50: 180nMAssay Description:Antagonist activity at HTR2C in human U2OS cells by PathHunter beta-arrestin assayMore data for this Ligand-Target Pair
Affinity DataIC50: 459nMAssay Description:Antagonist activity at human AVPR2 by PathHunter beta-arrestin assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.16E+3nMAssay Description:Antagonist activity at human OXTR expressed in CHO-K1 cells by PathHunter beta-arrestin assayMore data for this Ligand-Target Pair
TargetProlactin-releasing peptide receptor(Homo sapiens (Human))
University Of Florida
Curated by ChEMBL
University Of Florida
Curated by ChEMBL
Affinity DataIC50: 4.89E+3nMAssay Description:Antagonist activity at human PRLHR expressed in CHO-K1 cells by PathHunter beta-arrestin assayMore data for this Ligand-Target Pair
Affinity DataIC50: 7.29E+3nMAssay Description:Antagonist activity at human CCR8 expressed in CHO-K1 cells by PathHunter beta-arrestin assayMore data for this Ligand-Target Pair
Affinity DataIC50: 7.94E+3nMAssay Description:Antagonist activity at human CXCR4 expressed in mouse C2C12 cells by PathHunter beta-arrestin assayMore data for this Ligand-Target Pair
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
University Of Florida
Curated by ChEMBL
University Of Florida
Curated by ChEMBL
Affinity DataIC50: 8.03E+3nMAssay Description:Antagonist activity at human FSHR expressed in CHO-K1 cells by PathHunter beta-arrestin assayMore data for this Ligand-Target Pair
Affinity DataIC50: 8.30E+3nMAssay Description:Antagonist activity at human CCR3 expressed in CHO-K1 cells by PathHunter beta-arrestin assayMore data for this Ligand-Target Pair
Affinity DataIC50: 8.47E+3nMAssay Description:Antagonist activity at human CX3CR1 expressed in CHO-K1 cells by PathHunter beta-arrestin assayMore data for this Ligand-Target Pair