Compile Data Set for Download or QSAR
maximum 50k data
Found 11 Enz. Inhib. hit(s) with all data for entry = 50012751
TargetVasopressin V2 receptor(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM35723(CHEMBL344159 | N-[4-(7-Chloro-5-hydroxy-2,3,4,5-te...)
Affinity DataIC50:  0.00700nMAssay Description:Antagonist activity at human AVPR2 by PathHunter beta-arrestin assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50559938(CHEMBL154668)
Affinity DataIC50:  4.60nMAssay Description:Antagonist activity at human OXTR expressed in CHO-K1 cells by PathHunter beta-arrestin assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50559936(CHEMBL4744046)
Affinity DataIC50:  180nMAssay Description:Antagonist activity at HTR2C in human U2OS cells by PathHunter beta-arrestin assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetVasopressin V2 receptor(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50559937(CHEMBL4758081)
Affinity DataIC50:  459nMAssay Description:Antagonist activity at human AVPR2 by PathHunter beta-arrestin assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetOxytocin receptor(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50559937(CHEMBL4758081)
Affinity DataIC50:  1.16E+3nMAssay Description:Antagonist activity at human OXTR expressed in CHO-K1 cells by PathHunter beta-arrestin assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProlactin-releasing peptide receptor(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50559935(CHEMBL4780505)
Affinity DataIC50:  4.89E+3nMAssay Description:Antagonist activity at human PRLHR expressed in CHO-K1 cells by PathHunter beta-arrestin assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 8(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50559936(CHEMBL4744046)
Affinity DataIC50:  7.29E+3nMAssay Description:Antagonist activity at human CCR8 expressed in CHO-K1 cells by PathHunter beta-arrestin assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50559936(CHEMBL4744046)
Affinity DataIC50:  7.94E+3nMAssay Description:Antagonist activity at human CXCR4 expressed in mouse C2C12 cells by PathHunter beta-arrestin assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50559935(CHEMBL4780505)
Affinity DataIC50:  8.03E+3nMAssay Description:Antagonist activity at human FSHR expressed in CHO-K1 cells by PathHunter beta-arrestin assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 3(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50559936(CHEMBL4744046)
Affinity DataIC50:  8.30E+3nMAssay Description:Antagonist activity at human CCR3 expressed in CHO-K1 cells by PathHunter beta-arrestin assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCX3C chemokine receptor 1(Homo sapiens (Human))
University Of Florida

Curated by ChEMBL
LigandPNGBDBM50559936(CHEMBL4744046)
Affinity DataIC50:  8.47E+3nMAssay Description:Antagonist activity at human CX3CR1 expressed in CHO-K1 cells by PathHunter beta-arrestin assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed