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Found 8 Enz. Inhib. hit(s) with all data for entry = 50019101
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)TBA
LigandPNGBDBM50615252(CHEMBL5268610)
Affinity DataIC50:  1.31E+3nMAssay Description:Inhibition of HIV-1 reverse transcriptaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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Target15-hydroxyprostaglandin dehydrogenase [NAD(+)](Homo sapiens (Human))TBA
LigandPNGBDBM50103636(ADD-3878 | CHEBI:64227 | Ciglitazone | U-63287)
Affinity DataIC50:  2.70E+3nMAssay Description:Antagonist activity at 15-PGDH (unknown origin)More data for this Ligand-Target Pair
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LigandPNGBDBM50030474(Avandamet | Avandaryl | Avandia | BRL-49653 | CHEB...)
Affinity DataEC50:  730nMAssay Description:Agonist activity at GAL4-fused human PPARgamma expressed in HepG2 cellsMore data for this Ligand-Target Pair
LigandPNGBDBM50615253(CHEMBL5278539)
Affinity DataEC50:  10nMAssay Description:Agonist activity at human adrenergic receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetBeta-2 adrenergic receptor(Homo sapiens (Human))TBA
LigandPNGBDBM25763(5-[(2R)-2-{[(2R)-2-(3-chlorophenyl)-2-hydroxyethyl...)
Affinity DataEC50:  1.15E+3nMAssay Description:Agonist activity at human adrenergic receptor expressed in CHO cellsMore data for this Ligand-Target Pair
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LigandPNGBDBM50615250(CHEMBL5284791)
Affinity DataEC50:  284nMAssay Description:Agonist activity at human PPARgamma transfected in HEK293 cells assessed increase in luciferase activity incubated for 24 hrsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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LigandPNGBDBM50030474(Avandamet | Avandaryl | Avandia | BRL-49653 | CHEB...)
Affinity DataEC50:  9nMAssay Description:Agonist activity at human PPARgamma transfected in HEK293 cells assessed increase in luciferase activity incubated for 24 hrsMore data for this Ligand-Target Pair
LigandPNGBDBM50615251(CHEMBL5272825)
Affinity DataEC50:  190nMAssay Description:Agonist activity at GAL4-fused human PPARgamma expressed in HepG2 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed