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Found
1
Enz. Inhib. hit(s) with Target = 'Beta-lactamase TEM' and Ligand = 'BDBM466985'
Target
Beta-lactamase TEM
(Escherichia coli)
Entasis Therapeutics
US Patent
Ligand
BDBM466985
((2S)-2-fluoro-2-[[(2S,5R)-3-methyl-7-oxo-2-(pyrazi...)
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Affinity Data
IC50: 180nM
Assay Description:
A buffer consisting of 0.1 M sodium phosphate (pH 7.0), 10 mM NaHCO3, and 0.005% Triton X-100 was used for all enzymes. The chromogenic substrate nit...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
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Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
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