TargetCasein kinase I isoform gamma-2(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataIC50: 1.37E+3nMAssay Description:Inhibition of human CK1gamma2 using KRRRAL[pS]VASLPGL as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetCasein kinase I isoform gamma-2(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataIC50: 3.07E+3nMAssay Description:Inhibition of human CK1gamma2 using KRRRAL[pS]VASLPGL as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetCasein kinase I isoform gamma-2(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 780nMAssay Description:Binding constant for CSNK1G2 kinase domainMore data for this Ligand-Target Pair
TargetCasein kinase I isoform gamma-2(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 1.40E+3nMAssay Description:Average Binding Constant for CSNK1G2; NA=Not Active at 10 uMMore data for this Ligand-Target Pair
TargetCasein kinase I isoform gamma-2(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 780nMAssay Description:Binding constant for full-length CSNK1G2More data for this Ligand-Target Pair