Affinity DataKi: 2.70nMAssay Description:Inhibition of ERalpha in human MCF7 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 80nMAssay Description:Antagonist activity at human ERalpha receptor expressed in HEC1 cells assessed as transcriptional activation after 24 hrs by luciferase reporter gene...More data for this Ligand-Target Pair