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Found 2 Enz. Inhib. hit(s) with Target = 'Estrogen receptor' and Ligand = 'BDBM50254908'
TargetEstrogen receptor(Homo sapiens (Human))
Indian Institute Of Technology (Bhu)

Curated by ChEMBL
LigandPNGBDBM50254908(4-[1-(4-hydroxyphenyl)-4-methyl-5-{4-[2-(piperidin...)
Affinity DataKi:  2.70nMAssay Description:Inhibition of ERalpha in human MCF7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Indian Institute Of Technology (Bhu)

Curated by ChEMBL
LigandPNGBDBM50254908(4-[1-(4-hydroxyphenyl)-4-methyl-5-{4-[2-(piperidin...)
Affinity DataIC50:  80nMAssay Description:Antagonist activity at human ERalpha receptor expressed in HEC1 cells assessed as transcriptional activation after 24 hrs by luciferase reporter gene...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed