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Found 2 Enz. Inhib. hit(s) with Target = 'Histamine H3 receptor' and Ligand = 'BDBM50343849'
TargetHistamine H3 receptor(Homo sapiens (Human))
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50343849(3-(1H-Imidazol-4-yl)propylbut-3-enylcarbamate hydr...)
Affinity DataKi:  55nMAssay Description:Displacement of [125I]iodoproxyfan from human histamine H3 receptor expressed in CHO-K1 cells after 60 mins by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(GUINEA PIG)
Jagiellonian University Medical College

Curated by ChEMBL
LigandPNGBDBM50343849(3-(1H-Imidazol-4-yl)propylbut-3-enylcarbamate hydr...)
Affinity DataIC50:  68nMAssay Description:Antagonist activity against histamine H3 receptor in guinea pig ileum assessed as inhibition of electrically-evoked twitches after 30 mins in presenc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed