Compile Data Set for Download or QSAR
maximum 50k data
Found 5 Enz. Inhib. hit(s) with Target = 'Integrase' and Ligand = 'BDBM50237839'
TargetIntegrase(Human immunodeficiency virus 1)
Universit£

Curated by ChEMBL
LigandPNGBDBM50237839((R)-3-(4,5-dihydroxy-2-nitrophenyl)-2-(3-(3,4-dihy...)
Affinity DataIC50:  26nMAssay Description:Inhibition of HIV1 integrase using labelled U5A/U5B double stranded DNA substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Universit£

Curated by ChEMBL
LigandPNGBDBM50237839((R)-3-(4,5-dihydroxy-2-nitrophenyl)-2-(3-(3,4-dihy...)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of HIV1 integrase using labelled oligonucleotide substrate by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Universit£

Curated by ChEMBL
LigandPNGBDBM50237839((R)-3-(4,5-dihydroxy-2-nitrophenyl)-2-(3-(3,4-dihy...)
Affinity DataIC50:  3.70E+3nMAssay Description:Inhibition of HIV1 integrase strand transfer activity using labelled oligonucleotide substrate by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Universit£

Curated by ChEMBL
LigandPNGBDBM50237839((R)-3-(4,5-dihydroxy-2-nitrophenyl)-2-(3-(3,4-dihy...)
Affinity DataIC50:  5.47E+4nMAssay Description:Inhibition of HIV1 integrase using labelled oligonucleotide substrate in presence of bovine serum albumin by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Universit£

Curated by ChEMBL
LigandPNGBDBM50237839((R)-3-(4,5-dihydroxy-2-nitrophenyl)-2-(3-(3,4-dihy...)
Affinity DataIC50: >2.47E+5nMAssay Description:Inhibition of HIV1 integrase 3'-processing activity using labelled oligonucleotide substrate by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed