Compile Data Set for Download or QSAR
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Found 4 Enz. Inhib. hit(s) with Target = 'Kappa-type opioid receptor' and Ligand = 'BDBM50090002'
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50090002(CHEMBL411003 | Dynorphin A (1-11)-NH2H-Tyr-Gly-Gly...)
Affinity DataKi:  0.0590nMAssay Description:In vitro binding affinity towards human Opioid receptor kappa 1 on CHO cell membranes using [3H]diprenorphine displacement.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50090002(CHEMBL411003 | Dynorphin A (1-11)-NH2H-Tyr-Gly-Gly...)
Affinity DataKi:  0.0740nMAssay Description:Binding affinity towards cloned human Opioid receptor kappa 1 in CHO cell membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50090002(CHEMBL411003 | Dynorphin A (1-11)-NH2H-Tyr-Gly-Gly...)
Affinity DataEC50:  0.740nMAssay Description:Human kOpioid receptor kappa 1 mediated stimulation of [35S]- GTPgammaS binding in CHO cells (Agonist potency).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50090002(CHEMBL411003 | Dynorphin A (1-11)-NH2H-Tyr-Gly-Gly...)
Affinity DataEC50:  0.740nMAssay Description:Effective concentration for half-maximal stimulation was determined by [35S]GTP-gamma-S, assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed