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Found 4 Enz. Inhib. hit(s) with Target = 'Lethal(3)malignant brain tumor-like protein 3' and Ligand = 'BDBM50341828'
TargetLethal(3)malignant brain tumor-like protein 3(Homo sapiens (Human))
University of North Carolina

Curated by ChEMBL
LigandPNGBDBM50341828(3-bromo-5-[(4-pyrrolidin-1-ylpiperidin-1-yl)carbon...)
Affinity DataIC50:  2.80E+3nMAssay Description:Inhibition of His-tagged L3MBTL3 (unknown origin) using H4K20Me2 as substrate incubated for 30 mins at room temperature followed by incubation under ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLethal(3)malignant brain tumor-like protein 3(Homo sapiens (Human))
University of North Carolina

Curated by ChEMBL
LigandPNGBDBM50341828(3-bromo-5-[(4-pyrrolidin-1-ylpiperidin-1-yl)carbon...)
Affinity DataIC50:  3.10E+3nMAssay Description:Inhibition of L3MBTL3 (unknown origin) after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLethal(3)malignant brain tumor-like protein 3(Homo sapiens (Human))
University of North Carolina

Curated by ChEMBL
LigandPNGBDBM50341828(3-bromo-5-[(4-pyrrolidin-1-ylpiperidin-1-yl)carbon...)
Affinity DataIC50:  4.70E+3nMAssay Description:Inhibition of L3MBTL3 (unknown origin) using H4K20me2 as substrate after 30 mins by LNCE-TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLethal(3)malignant brain tumor-like protein 3(Homo sapiens (Human))
University of North Carolina

Curated by ChEMBL
LigandPNGBDBM50341828(3-bromo-5-[(4-pyrrolidin-1-ylpiperidin-1-yl)carbon...)
Affinity DataIC50:  3.50E+4nMAssay Description:Binding affinity to L3MBTL3 by chemiluminescent assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed