Found 2 Enz. Inhib. hit(s) with Target = 'Metabotropic glutamate receptor 2/3' and Ligand = 'BDBM50056272'
Affinity DataKi: 476nMAssay Description:Displacement of [3H]-LY459477 from mGlu2/3 receptor in Sprague-Dawley rat forebrain primary cortical membranes after 90 mins by liquid scintillation ...More data for this Ligand-Target Pair
Affinity DataEC50: 9.80nMAssay Description:Agonist activity at mGlu2/3 receptor in Sprague-Dawley rat forebrain assessed as inhibition of spontaneous Ca2+ oscillations in cortical neurons afte...More data for this Ligand-Target Pair