Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) with Target = 'Peroxisome proliferator-activated receptor gamma' and Ligand = 'BDBM50383922'
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Korea Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50383922(AMORPHASTILBOL)
Affinity DataIC50:  850nMAssay Description:Binding affinity to GST-tagged human PPARgamma by TR-FRET analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Korea Institute Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50383922(AMORPHASTILBOL)
Affinity DataEC50:  5.00E+3nMAssay Description:Transactivation of human PPARgamma expressed in african green monkey CV1 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed