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Found 4 Enz. Inhib. hit(s) with Target = 'Ras-related C3 botulinum toxin substrate 1' and Ligand = 'BDBM54568'
LigandPNGBDBM54568(1-[4-(2,5-dimethylphenyl)-1-piperazinyl]-3-[3-[2-(...)
Affinity DataKi:  200nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
LigandPNGBDBM54568(1-[4-(2,5-dimethylphenyl)-1-piperazinyl]-3-[3-[2-(...)
Affinity DataKi:  250nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
LigandPNGBDBM54568(1-[4-(2,5-dimethylphenyl)-1-piperazinyl]-3-[3-[2-(...)
Affinity DataEC50:  2.11E+3nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
LigandPNGBDBM54568(1-[4-(2,5-dimethylphenyl)-1-piperazinyl]-3-[3-[2-(...)
Affinity DataEC50:  2.70E+3nMAssay Description:University of New Mexico Assay Overview: Assay Support: NIH I RO3 MH081231-01 HTS to identify specific small molecule inhibitors of Ras and Ras-rela...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay