Found 3 Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein kinase 17A' and Ligand = 'BDBM50509365'
TargetSerine/threonine-protein kinase 17A(Homo sapiens (Human))
Uit - The Arctic University of Norway
Curated by ChEMBL
Uit - The Arctic University of Norway
Curated by ChEMBL
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of DRAK1 (unknown origin) expressed in HEK293 cells by NanoLuc-luciferase reporter based intracellular ATP competitiveness assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase 17A(Homo sapiens (Human))
Uit - The Arctic University of Norway
Curated by ChEMBL
Uit - The Arctic University of Norway
Curated by ChEMBL
Affinity DataIC50: 4.60E+3nMAssay Description:Inhibition of Alexa Fluor 647-labeled ATP competitive kinase tracer binding to GST-tagged DRAK1 (unknown origin) by FRET based cell free ATP-competit...More data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase 17A(Homo sapiens (Human))
Uit - The Arctic University of Norway
Curated by ChEMBL
Uit - The Arctic University of Norway
Curated by ChEMBL
Affinity DataKd: 2.80E+3nMAssay Description:Binding affinity to wild-type human partial length DRAK1 (R32 to E363 residues) expressed in bacterial expression system by active-site directed comp...More data for this Ligand-Target Pair