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Found 3 Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein kinase 17A' and Ligand = 'BDBM50509365'
TargetSerine/threonine-protein kinase 17A(Homo sapiens (Human))
Uit - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509365(CHEMBL4564337)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of DRAK1 (unknown origin) expressed in HEK293 cells by NanoLuc-luciferase reporter based intracellular ATP competitiveness assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase 17A(Homo sapiens (Human))
Uit - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509365(CHEMBL4564337)
Affinity DataIC50:  4.60E+3nMAssay Description:Inhibition of Alexa Fluor 647-labeled ATP competitive kinase tracer binding to GST-tagged DRAK1 (unknown origin) by FRET based cell free ATP-competit...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase 17A(Homo sapiens (Human))
Uit - The Arctic University of Norway

Curated by ChEMBL
LigandPNGBDBM50509365(CHEMBL4564337)
Affinity DataKd:  2.80E+3nMAssay Description:Binding affinity to wild-type human partial length DRAK1 (R32 to E363 residues) expressed in bacterial expression system by active-site directed comp...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed