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Found 3 Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein kinase PknB' and Ligand = 'BDBM50421679'
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)TBA
LigandPNGBDBM50421679(CHEMBL5282708)
Affinity DataKi:  440nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant PknB (1 to 331 residues) expressed in Escherichia coli BL21-Rosetta cells using GarA and ATP as ...More data for this Ligand-Target Pair
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TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)TBA
LigandPNGBDBM50421679(CHEMBL5282708)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant PknB (1 to 331 residues) expressed in Escherichia coli BL21-Rosetta cells using GarA and ATP as ...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)TBA
LigandPNGBDBM50421679(CHEMBL5282708)
Affinity DataKd:  30nMAssay Description:Binding affinity to Mycobacterium tuberculosis recombinant N-terminal His-tagged PknB (1 to 331 residues) expressed in Escherichia coli DH5alpha cell...More data for this Ligand-Target Pair
In DepthDetails PubMed