Compile Data Set for Download or QSAR
maximum 50k data
Found 3 Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein kinase PknB' and Ligand = 'BDBM50421684'
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)TBA
LigandPNGBDBM50421684(CHEMBL5277619)
Affinity DataKi:  1.90E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant PknB (1 to 331 residues) expressed in Escherichia coli BL21-Rosetta cells using GarA and ATP as ...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)TBA
LigandPNGBDBM50421684(CHEMBL5277619)
Affinity DataIC50:  6.60E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant PknB (1 to 331 residues) expressed in Escherichia coli BL21-Rosetta cells using GarA and ATP as ...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)TBA
LigandPNGBDBM50421684(CHEMBL5277619)
Affinity DataKd:  660nMAssay Description:Binding affinity to Mycobacterium tuberculosis recombinant N-terminal His-tagged PknB (1 to 331 residues) expressed in Escherichia coli DH5alpha cell...More data for this Ligand-Target Pair
In DepthDetails PubMed