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Found 4 Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein kinase PknB' and Ligand = 'BDBM50421686'
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)TBA
LigandPNGBDBM50421686(CHEMBL5282194)
Affinity DataKi:  320nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant PknB (1 to 331 residues) expressed in Escherichia coli BL21-Rosetta cells using GarA and ATP as ...More data for this Ligand-Target Pair
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TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)TBA
LigandPNGBDBM50421686(CHEMBL5282194)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis recombinant PknB (1 to 331 residues) expressed in Escherichia coli BL21-Rosetta cells using GarA and ATP as ...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)TBA
LigandPNGBDBM50421686(CHEMBL5282194)
Affinity DataKd:  34nMAssay Description:Binding affinity to Mycobacterium tuberculosis recombinant N-terminal His-tagged PknB (1 to 331 residues) expressed in Escherichia coli DH5alpha cell...More data for this Ligand-Target Pair
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TargetSerine/threonine-protein kinase PknB(Mycobacterium tuberculosis)TBA
LigandPNGBDBM50421686(CHEMBL5282194)
Affinity DataKd:  19nMAssay Description:Binding affinity to Mycobacterium tuberculosis partial length PknB (M1 to G279 residues) expressed in mammalian expression system by KdELECT kinase a...More data for this Ligand-Target Pair
In DepthDetails PubMed