Found 2 Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein kinase pim-3' and Ligand = 'BDBM50509365'
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Uit - The Arctic University of Norway
Curated by ChEMBL
Uit - The Arctic University of Norway
Curated by ChEMBL
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of PIM3 (unknown origin) by [33P]-ATP filter binding kinase assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Uit - The Arctic University of Norway
Curated by ChEMBL
Uit - The Arctic University of Norway
Curated by ChEMBL
Affinity DataKd: 4.70E+3nMAssay Description:Binding affinity to wild-type human partial length PIM3 (G16 to A317 residues) expressed in bacterial expression system by active-site directed compe...More data for this Ligand-Target Pair