Compile Data Set for Download or QSAR
maximum 50k data
Found 4 Enz. Inhib. hit(s) with Target = 'Thromboxane A2 receptor' and Ligand = 'BDBM50353634'
TargetThromboxane A2 receptor(MOUSE)
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50353634(CHEMBL1828642)
Affinity DataIC50:  1.63E+3nMAssay Description:Antagonist activity at mouse prostanoid TP receptor expressed in QBI-HEK 293A cells assessed as inhibition of 1-BOP-induced increase in inositol mono...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50353634(CHEMBL1828642)
Affinity DataIC50:  1.51E+4nMAssay Description:Antagonist activity at human prostanoid TP receptor expressed in QBI-HEK 293A cells assessed as inhibition of 1-BOP-induced increase in inositol mono...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50353634(CHEMBL1828642)
Affinity DataKd: >1.00E+4nMAssay Description:Displacement of [3H]SQ-29548 from human prostanoid TP receptor expressed in QBI-HEK 293A cells after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(MOUSE)
University Of Pennsylvania

Curated by ChEMBL
LigandPNGBDBM50353634(CHEMBL1828642)
Affinity DataKd:  1.00E+4nMAssay Description:Displacement of [3H]SQ-29548 from mouse prostanoid TP receptor expressed in QBI-HEK 293A cells after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed