Found 5 Enz. Inhib. hit(s) with Target = 'Type-1 angiotensin II receptor' and Ligand = 'BDBM50047126'
Affinity DataIC50: 5nMAssay Description:In vitro antagonistic potency against Angiotensin II receptor, type 1 in guinea pig adrenal membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Compound was tested for in vitro inhibition of specific binding of [I-125]AII to Angiotensin II receptor, type 1 in guinea pig adrenal membrane prepa...More data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Binding affinity to angiotensin AT1 receptor in guinea pig adrenal cortex membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Inhibition of [125I]-Angiotensin binding to a guinea pig adrenal membrane preparation which corresponds to Angiotensin II receptor, type 1More data for this Ligand-Target Pair
Affinity DataKd: 0.0501nMAssay Description:Antagonist activity at angiotensin AT1 receptor in rabbit aortaMore data for this Ligand-Target Pair