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Found 15 Enz. Inhib. hit(s) with all data for assayid = 2 entry = 50005942
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50001462(3-[(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylam...)
Affinity DataKi:  56nMAssay Description:Binding affinity was determined on mu [3H]-DAGO site in rat brain synaptosomes by radioreceptor assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50042763(CHEMBL263698 | H-Tyr-D-Ala-deltaPhe-Asp-Val-Val-Gl...)
Affinity DataKi:  114nMAssay Description:Binding affinity was determined on mu [3H]-DAGO site in rat brain synaptosomes by radioreceptor assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50001459(3-[(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylam...)
Affinity DataKi:  178nMAssay Description:Binding affinity was determined on mu [3H]-DAGO site in rat brain synaptosomes by radioreceptor assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50001468((S)-3-((S)-2-{(R)-2-[(S)-2-Amino-3-(4-hydroxy-phen...)
Affinity DataKi:  205nMAssay Description:Binding affinity was determined on mu [3H]-DAGO site in rat brain synaptosomes by radioreceptor assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50042762(CHEMBL339456 | H-Tyr-D-Ala-Nap(1)-Asp-Val-Val-Gly-...)
Affinity DataKi:  279nMAssay Description:Binding affinity was determined on mu [3H]-DAGO site in rat brain synaptosomes by radioreceptor assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50042766(CHEMBL125872 | H-Tyr-D-Ala-Trp-Asp-Val-Val-Gly-NH2)
Affinity DataKi:  323nMAssay Description:Binding affinity was determined on mu [3H]-DAGO site in rat brain synaptosomes by radioreceptor assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50042769(CHEMBL332416 | H-Tyr-D-Ala-Hfe-Asp-Val-Val-Gly-NH2)
Affinity DataKi:  326nMAssay Description:Binding affinity was determined on mu [3H]-DAGO site in rat brain synaptosomes by radioreceptor assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50042764(CHEMBL339683 | H-Tyr-D-Ala-Tyr(OMe)-Asp-Val-Val-Gl...)
Affinity DataKi:  526nMAssay Description:Binding affinity was determined on mu [3H]-DAGO site in rat brain synaptosomes by radioreceptor assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50042768(CHEMBL125285 | H-Tyr-D-Ala-Nap(2)-Asp-Val-Val-Gly-...)
Affinity DataKi:  770nMAssay Description:Binding affinity was determined on mu [3H]-DAGO site in rat brain synaptosomes by radioreceptor assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50042767(CHEMBL334299 | H-Tyr-D-Ala-Tyr-Asp-Val-Val-Gly-NH2)
Affinity DataKi:  1.18E+3nMAssay Description:Binding affinity was determined on mu [3H]-DAGO site in rat brain synaptosomes by radioreceptor assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50042760(CHEMBL121946 | H-Tyr-D-Ala-(R or S)CalphaMPhe-Asp-...)
Affinity DataKi:  1.36E+3nMAssay Description:Binding affinity was determined on mu [3H]-DAGO site in rat brain synaptosomes by radioreceptor assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50042759(CHEMBL125289 | H-Tyr-D-Ala-His-Asp-Val-Val-Gly-NH2)
Affinity DataKi:  3.72E+3nMAssay Description:Binding affinity was determined on mu [3H]-DAGO site in rat brain synaptosomes by radioreceptor assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50042761(CHEMBL340909 | H-Tyr-D-Ala-Phg-Asp-Val-Val-Gly-NH2)
Affinity DataKi:  3.75E+3nMAssay Description:Binding affinity was determined on mu [3H]-DAGO site in rat brain synaptosomes by radioreceptor assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50001460(3-[(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylam...)
Affinity DataKi:  7.81E+3nMAssay Description:Binding affinity was determined on mu [3H]-DAGO site in rat brain synaptosomes by radioreceptor assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University of Ferrara

Curated by ChEMBL
LigandPNGBDBM50042765(CHEMBL122159 | H-Tyr-D-Ala-NalphaMePhe-Asp-Val-Val...)
Affinity DataKi:  1.90E+4nMAssay Description:Binding affinity was determined on mu [3H]-DAGO site in rat brain synaptosomes by radioreceptor assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed