Compile Data Set for Download or QSAR
maximum 50k data
Found 8 Enz. Inhib. hit(s) with all data for assayid = 2 entry = 50010100
TargetProtein-arginine deiminase type-4(Homo sapiens (Human))
Yale University

Curated by ChEMBL
LigandPNGBDBM50535207(CHEMBL4449566)
Affinity DataIC50:  8.80E+3nMAssay Description:Inhibition of recombinant human GST-tagged PAD4 expressed in Escherichia coli BL21-DE3 pLysS assessed as reduction in reduction in residual activity ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-arginine deiminase type-4(Homo sapiens (Human))
Yale University

Curated by ChEMBL
LigandPNGBDBM50535208(CHEMBL4547728)
Affinity DataIC50:  2.20E+4nMAssay Description:Inhibition of recombinant human GST-tagged PAD4 expressed in Escherichia coli BL21-DE3 pLysS assessed as reduction in reduction in residual activity ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-arginine deiminase type-4(Homo sapiens (Human))
Yale University

Curated by ChEMBL
LigandPNGBDBM50535204(CHEMBL4468883)
Affinity DataIC50:  2.80E+4nMAssay Description:Inhibition of recombinant human GST-tagged PAD4 expressed in Escherichia coli BL21-DE3 pLysS assessed as reduction in reduction in residual activity ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-arginine deiminase type-4(Homo sapiens (Human))
Yale University

Curated by ChEMBL
LigandPNGBDBM50535201(CHEMBL4442207)
Affinity DataIC50:  3.60E+4nMAssay Description:Inhibition of recombinant human GST-tagged PAD4 expressed in Escherichia coli BL21-DE3 pLysS assessed as reduction in reduction in residual activity ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-arginine deiminase type-4(Homo sapiens (Human))
Yale University

Curated by ChEMBL
LigandPNGBDBM50535206(CHEMBL4464539)
Affinity DataIC50:  3.90E+4nMAssay Description:Inhibition of recombinant human GST-tagged PAD4 expressed in Escherichia coli BL21-DE3 pLysS assessed as reduction in reduction in residual activity ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-arginine deiminase type-4(Homo sapiens (Human))
Yale University

Curated by ChEMBL
LigandPNGBDBM50535203(CHEMBL4473416)
Affinity DataIC50:  5.30E+4nMAssay Description:Inhibition of recombinant human GST-tagged PAD4 expressed in Escherichia coli BL21-DE3 pLysS assessed as reduction in reduction in residual activity ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-arginine deiminase type-4(Homo sapiens (Human))
Yale University

Curated by ChEMBL
LigandPNGBDBM50535202(CHEMBL4546087)
Affinity DataIC50:  6.40E+4nMAssay Description:Inhibition of recombinant human GST-tagged PAD4 expressed in Escherichia coli BL21-DE3 pLysS assessed as reduction in reduction in residual activity ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein-arginine deiminase type-4(Homo sapiens (Human))
Yale University

Curated by ChEMBL
LigandPNGBDBM50535205(CHEMBL4461562)
Affinity DataIC50:  1.29E+5nMAssay Description:Inhibition of recombinant human GST-tagged PAD4 expressed in Escherichia coli BL21-DE3 pLysS assessed as reduction in reduction in residual activity ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed