Compile Data Set for Download or QSAR
maximum 50k data
Found 477 of ic50 for UniProtKB: P35351
LigandPNGBDBM50030815(CHEMBL404594)
Affinity DataIC50:  0.100nMAssay Description:Binding affinity for rat brain Angiotensin II receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50230790(CHEMBL292892)
Affinity DataIC50:  0.150nMAssay Description:Inhibition of [125I]AII binding to Angiotensin II receptor, type 1 of rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50230779(CHEMBL294686)
Affinity DataIC50:  0.300nMAssay Description:Inhibition of [125I]AII binding to Angiotensin II receptor, type 1 of rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50030815(CHEMBL404594)
Affinity DataIC50:  0.350nMAssay Description:Binding affinity against Angiotensin II receptor, from rat adrenal glandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50230811(CHEMBL293091)
Affinity DataIC50:  0.400nMAssay Description:Inhibition of [125I]AII binding to Angiotensin II receptor, type 1 of rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50230778(CHEMBL56211)
Affinity DataIC50:  0.560nMAssay Description:Inhibition of [125I]AII binding to Angiotensin II receptor, type 1 of rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50230771(CHEMBL55510)
Affinity DataIC50:  0.590nMAssay Description:Inhibition of [125I]AII binding to Angiotensin II receptor, type 1 of rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50230806(CHEMBL294415)
Affinity DataIC50:  0.800nMAssay Description:Inhibition of [125I]AII binding to Angiotensin II receptor, type 1 of rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50048078(4-[2-Butyl-5-((E)-2-carboxy-3-thiophen-2-yl-propen...)
Affinity DataIC50:  1nMAssay Description:Inhibition of [125I]AII binding to Angiotensin II receptor, type 1 of rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50212829(CHEMBL170944)
Affinity DataIC50:  1.20nMAssay Description:Angiotensin II receptor antagonist activity was determined by 50% inhibition of specific binding of [3H]angiotensin II (2 nM) to rat adrenal cortical...More data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50042235(2-butyl-3-{[2'-(1H-tetrazol-5-yl)[1,1'-biphenyl]-4...)
Affinity DataIC50:  1.30nMAssay Description:Inhibition of [125I]-AII binding to Angiotensin II receptor of rat uterine membraneMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50228195(Angiotensin Ii | CHEBI:2719)
Affinity DataIC50:  1.30nMAssay Description:Binding affinity against Angiotensin II receptor, from rat adrenal glandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50011975(4-[2-Butyl-5-((E)-2-carboxy-3-thiophen-2-yl-propen...)
Affinity DataIC50:  1.5nMAssay Description:Inhibition of [125I]AII binding to Angiotensin II receptor, type 1 of rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228894(CHEMBL312754)
Affinity DataIC50:  1.60nMAssay Description:Binding affinity against Angiotensin II receptor, from rat adrenal glandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50236697(5-L-isoleucineangiotensin II | 5-isoleucine-angiot...)
Affinity DataIC50:  2nMAssay Description:Angiotensin II receptor antagonist activity was determined by 50% inhibition of specific binding of [3H]angiotensin II (2 nM) to rat adrenal cortical...More data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50281848(2-Ethyl-5,7-dimethyl-3-{4-[2-(2H-tetrazol-5-yl)-5H...)
Affinity DataIC50:  2.30nMAssay Description:Compound was tested for inhibition of Angiotensin II receptor in rabbit aorta binding assayMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50212853(CHEMBL274626)
Affinity DataIC50:  2.40nMAssay Description:Compound was tested for inhibition of Angiotensin II receptor in rabbit aorta binding assayMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50230787(CHEMBL54421)
Affinity DataIC50:  2.5nMAssay Description:Inhibition of [125I]AII binding to Angiotensin II receptor, type 1 of rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50212825(CHEMBL435855)
Affinity DataIC50:  3nMAssay Description:Competitive inhibition of Angiotensin II receptor binding of radiolabeled AII to rat adrenal glomerulosa tissue by 50%More data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50230792(CHEMBL56497)
Affinity DataIC50:  3.30nMAssay Description:Inhibition of [125I]AII binding to Angiotensin II receptor, type 1 of rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50230799(CHEMBL56333)
Affinity DataIC50:  3.30nMAssay Description:Inhibition of [125I]AII binding to Angiotensin II receptor, type 1 of rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50228195(Angiotensin Ii | CHEBI:2719)
Affinity DataIC50:  4nMAssay Description:Binding affinity for rat brain Angiotensin II receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50230774(CHEMBL291955)
Affinity DataIC50:  4.30nMAssay Description:Inhibition of [125I]AII binding to Angiotensin II receptor, type 1 of rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50230762(CHEMBL56160)
Affinity DataIC50:  4.5nMAssay Description:Inhibition of [125I]AII binding to Angiotensin II receptor, type 1 of rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50212843(CHEMBL267809)
Affinity DataIC50:  4.5nMAssay Description:Inhibition of [125I]-AII binding to Angiotensin II receptor of rat uterine membraneMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50230810(CHEMBL299064)
Affinity DataIC50:  4.60nMAssay Description:Inhibition of [125I]AII binding to Angiotensin II receptor, type 1 of rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM82258(CAS_114798-26-4 | Losartan | NSC_3961)
Affinity DataIC50:  4.60nMAssay Description:Displacement of [3H]-AII from the Angiotensin II receptor isolated from the liver of ratsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50230764(CHEMBL299954)
Affinity DataIC50:  4.80nMAssay Description:Inhibition of [125I]AII binding to Angiotensin II receptor, type 1 of rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50281823(4-Butyl-1-((1R,2R,6S)-2,6-dimethyl-cyclohexyl)-3-{...)
Affinity DataIC50:  4.90nMAssay Description:Inhibition of [125I]-AII binding to Angiotensin II receptor of rat uterine membraneMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50212845(CHEMBL274668)
Affinity DataIC50:  5nMAssay Description:Inhibition of [125I]-AII binding to Angiotensin II receptor of rat uterine membraneMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50212849(CHEMBL430152)
Affinity DataIC50:  5nMAssay Description:Inhibition of [125I]-AII binding to Angiotensin II receptor of rat uterine membraneMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50230767(CHEMBL56522)
Affinity DataIC50:  5nMAssay Description:Inhibition of [125I]AII binding to Angiotensin II receptor, type 1 of rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50212952(CHEMBL46150)
Affinity DataIC50:  5nMAssay Description:In vitro Angiotensin II receptor antagonist activity in rat adrenal cortex tissue.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50228894(CHEMBL312754)
Affinity DataIC50:  5.10nMAssay Description:Binding affinity for rat brain Angiotensin II receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50046078(5-[4'-(3,5-Dibutyl-[1,2,4]triazol-1-ylmethyl)-biph...)
Affinity DataIC50:  5.60nMAssay Description:Tested in vitro for inhibition of [125I]AII to rat uterine membranesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50046078(5-[4'-(3,5-Dibutyl-[1,2,4]triazol-1-ylmethyl)-biph...)
Affinity DataIC50:  5.60nMAssay Description:Inhibition of [125I]-AII binding to Angiotensin II receptor of rat uterine membraneMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50049207(2-Butyl-6-(1-methoxy-1-methyl-ethyl)-3-[2'-(1H-tet...)
Affinity DataIC50:  6nMAssay Description:In vitro Angiotensin II receptor antagonist activity in rat adrenal cortex tissue.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50212830(CHEMBL171524)
Affinity DataIC50:  6.40nMAssay Description:Angiotensin II receptor antagonist activity was determined by 50% inhibition of specific binding of [3H]angiotensin II (2 nM) to rat adrenal cortical...More data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50281814(1,4-Dibutyl-3-{6-[2-(1H-tetrazol-5-yl)-phenyl]-pyr...)
Affinity DataIC50:  6.5nMAssay Description:Inhibition of [125I]-AII binding to Angiotensin II receptor of rat uterine membraneMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50230796(CHEMBL56690)
Affinity DataIC50:  6.60nMAssay Description:Inhibition of [125I]AII binding to Angiotensin II receptor, type 1 of rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50145967(2-(3,5-Dibutyl-[1,2,4]triazol-1-ylmethyl)-5-[2-(1H...)
Affinity DataIC50:  6.80nMAssay Description:Tested in vitro for inhibition of [125I]AII to rat uterine membranesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50049209(5-(3,5-Dibutyl-[1,2,4]triazol-1-ylmethyl)-2-[2-(1H...)
Affinity DataIC50:  6.90nMAssay Description:Inhibition of [125I]-AII binding to Angiotensin II receptor of rat uterine membraneMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50049209(5-(3,5-Dibutyl-[1,2,4]triazol-1-ylmethyl)-2-[2-(1H...)
Affinity DataIC50:  6.90nMAssay Description:Tested in vitro for inhibition of [125I]AII to rat uterine membranesMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50212844(CHEMBL276689)
Affinity DataIC50:  9.40nMAssay Description:Inhibition of [125I]-AII binding to Angiotensin II receptor of rat uterine membraneMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50230772(CHEMBL59043)
Affinity DataIC50: >10nMAssay Description:Inhibition of [125I]AII binding to Angiotensin II receptor, type 1 of rat mesenteric arteriesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50212954(CHEMBL295114)
Affinity DataIC50:  11nMAssay Description:In vitro Angiotensin II receptor antagonist activity in rat adrenal cortex tissue.More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50281822(1,4-Dibutyl-3-[2'-(1H-tetrazol-5-yl)-biphenyl-4-yl...)
Affinity DataIC50:  12nMAssay Description:Inhibition of [125I]-AII binding to Angiotensin II receptor of rat uterine membraneMore data for this Ligand-Target Pair
In DepthDetails
LigandPNGBDBM50229469(CHEMBL315094)
Affinity DataIC50:  12nMAssay Description:Inhibition of radioligand [3H]angiotensin II binding to angiotensin II receptor of rat adrenal cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50226528(CHEMBL284425)
Affinity DataIC50:  12nMAssay Description:Inhibitory concentration that gave 50 percent displacement of specific binding of [3H]AII (2 nM) to Angiotensin II receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM82258(CAS_114798-26-4 | Losartan | NSC_3961)
Affinity DataIC50:  13nMAssay Description:Competitive inhibition of Angiotensin II receptor binding of radiolabeled AII to rat adrenal glomerulosa tissue by 50%More data for this Ligand-Target Pair
In DepthDetails
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