Compile Data Set for Download or QSAR
maximum 50k data
Found 3 of ic50 for monomerid = 50035444
TargetType-1 angiotensin II receptor(RABBIT)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50035444(4-[[2'-[N-(tert-Butoxycarbonyl)sulfamoyl]biphenyl-...)
Affinity DataIC50:  0.0720nMAssay Description:Tested for in vitro binding affinity against angiotensin I (AT1) receptor to competitively block the specific binding of [125I]- [Sar1,Ile8] AII to a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(RABBIT)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50035444(4-[[2'-[N-(tert-Butoxycarbonyl)sulfamoyl]biphenyl-...)
Affinity DataIC50:  0.0720nMAssay Description:Antagonist activity at AT1 receptor in rabbit aorta membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-2 angiotensin II receptor(RAT)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50035444(4-[[2'-[N-(tert-Butoxycarbonyl)sulfamoyl]biphenyl-...)
Affinity DataIC50:  1.40nMAssay Description:In vitro binding affinity against angiotensin II (AT2) receptor to competitively block the specific binding of [125I]- [Sar1,Ile8] AII to a rat mid b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed