Affinity DataIC50: 615nMAssay Description:Antagonist activity at human iGluA1 receptor flop isoform expressed in CHO-S cells coexpressing TARP gamma-8 and human EAAT3 assessed as inhibition o...More data for this Ligand-Target Pair
Affinity DataIC50: 4.67E+3nMAssay Description:Inhibition of human CYP1A2More data for this Ligand-Target Pair
Affinity DataIC50: 9.26E+3nMAssay Description:Antagonist activity at human iGluA1 receptor flip isoform expressed in CHO-S cells assessed as inhibition of glutamate-induced increase in intracellu...More data for this Ligand-Target Pair
Affinity DataIC50: 8.33E+4nMAssay Description:Antagonist activity at human iGluA1 receptor flop isoform expressed in CHO-S cells coexpressing TARP gamma-2 assessed as inhibition of glutamate-indu...More data for this Ligand-Target Pair