Affinity DataIC50: 1nMAssay Description:Displacement of [125I]glucagon from human GCGR expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Antagonist activity against human GCGR expressed in CHO cells assessed as glucagon-induced cAMP accumulationMore data for this Ligand-Target Pair
TargetGastric inhibitory polypeptide(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:Binding affinity against human GIPMore data for this Ligand-Target Pair
Affinity DataIC50: 5.00E+3nMAssay Description:Binding affinity against human GLP1More data for this Ligand-Target Pair