Compile Data Set for Download or QSAR
maximum 50k data
Found 4 of ic50 for monomerid = 50292977
TargetOrexin receptor type 2(Homo sapiens (Human))
Actelion Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50292977(2-(3,4-dimethoxy-N-p-tolylphenylsulfonamido)-N,N-d...)
Affinity DataIC50:  19nMAssay Description:Antagonist activity at OX2 receptor by FLIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin receptor type 2(Homo sapiens (Human))
Actelion Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50292977(2-(3,4-dimethoxy-N-p-tolylphenylsulfonamido)-N,N-d...)
Affinity DataIC50:  19nMAssay Description:Inhibition of human OX2 receptor expressed in CHO cells assessed as intercellular calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Actelion Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50292977(2-(3,4-dimethoxy-N-p-tolylphenylsulfonamido)-N,N-d...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human OX1 receptor expressed in CHO cells assessed as intercellular calcium mobilization by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetOrexin/Hypocretin receptor type 1(Homo sapiens (Human))
Actelion Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50292977(2-(3,4-dimethoxy-N-p-tolylphenylsulfonamido)-N,N-d...)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at OX1 receptor by FLIPRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed