Compile Data Set for Download or QSAR
maximum 50k data
Found 3 of ic50 for monomerid = 50343571
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
Nerviano Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50343571((S)-1-methyl-8-(5-(pyrrolidine-2-carboxamido)-2-(t...)
Affinity DataIC50:  44nMAssay Description:Inhibition of PLK1 assessed as [33P]gamma-ATP incorporation into substrate after 60 mins by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK3(Homo sapiens (Human))
Nerviano Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50343571((S)-1-methyl-8-(5-(pyrrolidine-2-carboxamido)-2-(t...)
Affinity DataIC50:  681nMAssay Description:Inhibition of PLK3 assessed as [33P]gamma-ATP incorporation into substrate after 60 mins by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK2(Homo sapiens (Human))
Nerviano Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50343571((S)-1-methyl-8-(5-(pyrrolidine-2-carboxamido)-2-(t...)
Affinity DataIC50:  1.45E+3nMAssay Description:Inhibition of PLK2 assessed as [33P]gamma-ATP incorporation into substrate after 60 mins by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed