Compile Data Set for Download or QSAR
maximum 50k data
Found 7 of ic50 for monomerid = 50379707
TargetP2X purinoceptor 3(Homo sapiens (Human))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50379707(CHEMBL2011112)
Affinity DataIC50:  20nMAssay Description:Antagonist activity at human P2X3 receptor expressed in HEK293 Flp-in cells assessed as inhibition of alpha-beta-methylene-ATP induced calcium releas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50379707(CHEMBL2011112)
Affinity DataIC50:  20nMAssay Description:Antagonist activity at human P2X3 receptor expressed in HEK293 Flp-in cells assessed as inhibition of alpha-beta-methylene-ATP induced calcium releas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50379707(CHEMBL2011112)
Affinity DataIC50:  25nMAssay Description:Antagonist activity at human recombinant P2X3 receptor expressed in HEK293-Tet-on cells assessed as alpha,beta-methylene-ATP-stimulated Ca2+ influx b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50379707(CHEMBL2011112)
Affinity DataIC50:  25nMAssay Description:Antagonist activity at human recombinant P2X3 receptor expressed in HEK293-Tet-on cells assessed as alpha,beta-methylene-ATP-stimulated Ca2+ influx b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(Homo sapiens (Human))
Gedeon Richter

Curated by ChEMBL
LigandPNGBDBM50379707(CHEMBL2011112)
Affinity DataIC50:  61nMAssay Description:Antagonist activity at human P2X3 receptor expressed in RLE cells assessed as inhibition of (alpha,beta)me-ATP-induced intracellular calcium level by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetP2X purinoceptor 3(RAT)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50379707(CHEMBL2011112)
Affinity DataIC50:  280nMAssay Description:Antagonist activity at rat P2X3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50379707(CHEMBL2011112)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of recombinant CYP2C9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed