TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Arizona
Curated by ChEMBL
University Of Arizona
Curated by ChEMBL
Affinity DataKi: 1.30nMAssay Description:Binding affinity towards Cholecystokinin type B receptor (CCK-B) receptor was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 1.5nM ΔG°: -50.4kJ/mole EC50: 23nMpH: 7.4 T: 2°CAssay Description:Log IC50 values for each test compound were determined from nonlinear regression analysis of data collected from two independent experiments performe...More data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
University Of Arizona
Curated by ChEMBL
University Of Arizona
Curated by ChEMBL
Affinity DataKi: 1.5nM EC50: 6.60nMAssay Description:Log IC50 values for each test compound were determined from nonlinear regression analysis of data collected from two independent experiments performe...More data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Binding affinity towards Opioid receptor delta 1 was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Binding affinity towards Opioid receptor mu 1 was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 22nM ΔG°: -43.7kJ/mole EC50: 38nMpH: 7.4 T: 2°CAssay Description:Log IC50 values for each test compound were determined from nonlinear regression analysis of data collected from two independent experiments performe...More data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Binding affinity towards Cholecystokinin type A receptor (CCK-A) receptor was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 320nMAssay Description:Log IC50 values for each test compound were determined from nonlinear regression analysis of data collected from two independent experiments performe...More data for this Ligand-Target Pair