Compile Data Set for Download or QSAR
maximum 50k data
Found 4 of ki for monomerid = 21381
Target5-hydroxytryptamine receptor 7(Rattus norvegicus (rat))
Universita Degli Studi Di Bari

LigandPNGBDBM21381(6-{4-[2-(propan-2-yl)phenyl]piperazin-1-yl}-N-(1,2...)
Affinity DataKi:  1.10nM ΔG°:  -53.2kJ/molepH: 7.4 T: 2°CAssay Description:IC50 values for each test compound were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibiti...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Universita Degli Studi Di Bari

LigandPNGBDBM21381(6-{4-[2-(propan-2-yl)phenyl]piperazin-1-yl}-N-(1,2...)
Affinity DataKi:  15nMAssay Description:IC50 values for each test compound were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibiti...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Universita Degli Studi Di Bari

LigandPNGBDBM21381(6-{4-[2-(propan-2-yl)phenyl]piperazin-1-yl}-N-(1,2...)
Affinity DataKi:  167nMAssay Description:IC50 values for each test compound were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibiti...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Universita Degli Studi Di Bari

LigandPNGBDBM21381(6-{4-[2-(propan-2-yl)phenyl]piperazin-1-yl}-N-(1,2...)
Affinity DataKi:  4.82E+3nMAssay Description:IC50 values for each test compound were determined from nonlinear regression analysis of data collected from ligand binding experiments. The inhibiti...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed