TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Zambeletti Research Laboratories
Curated by ChEMBL
Zambeletti Research Laboratories
Curated by ChEMBL
Affinity DataKi: 0.640nMAssay Description:Displacement of [3H]-BRL 52537 from opioid receptor kappa site in guinea pigMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Mus musculus (Mouse))
Smithkline Beecham Farmaceutici
Curated by ChEMBL
Smithkline Beecham Farmaceutici
Curated by ChEMBL
Affinity DataKi: 0.640nMAssay Description:Evaluated for the binding affinity at kappa receptorMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Zambeletti Research Laboratories
Curated by ChEMBL
Zambeletti Research Laboratories
Curated by ChEMBL
Affinity DataKi: 1.00E+3nMAssay Description:Binding affinity of the compound was measured on opioid receptor delta sites.More data for this Ligand-Target Pair
Affinity DataKi: 2.34E+3nMAssay Description:Affinity for opioid receptor mu sitesMore data for this Ligand-Target Pair