Compile Data Set for Download or QSAR
maximum 50k data
Found 5 of ki for monomerid = 50037483
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50037483((+)-cis-N-Normetazocine | (6S,11R)-6,11-Dimethyl-1...)
Affinity DataKi:  23nMAssay Description:Inhibition against mu receptor using [3H]DAMGO in homogenate of rat brain cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50037483((+)-cis-N-Normetazocine | (6S,11R)-6,11-Dimethyl-1...)
Affinity DataKi:  54nMAssay Description:Inhibition against mu receptor from displacement studies using 0.5 nM [3H]-DAMGO in rhesus monkey cortex membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50037483((+)-cis-N-Normetazocine | (6S,11R)-6,11-Dimethyl-1...)
Affinity DataKi:  113nMAssay Description:Inhibition against kappa receptor from displacement studies using 1.5 nM [3H]U-69593 in rhesus monkey cortex membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50037483((+)-cis-N-Normetazocine | (6S,11R)-6,11-Dimethyl-1...)
Affinity DataKi:  449nMAssay Description:Inhibition against delta receptor from displacement studies using 1.5 nM [3H]DPDPE in rhesus monkey cortex membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Virginia Commonwealth University

Curated by ChEMBL
LigandPNGBDBM50037483((+)-cis-N-Normetazocine | (6S,11R)-6,11-Dimethyl-1...)
Affinity DataKi:  6.75E+3nMAssay Description:Inhibition against sigma receptor using displacement of 3 nM [3H]pentazocine in homogenate of guinea pig brain cerebellumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed