TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
F. Hoffmann-La Roche
Curated by PDSP Ki Database
F. Hoffmann-La Roche
Curated by PDSP Ki Database
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
F. Hoffmann-La Roche
Curated by PDSP Ki Database
F. Hoffmann-La Roche
Curated by PDSP Ki Database
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
F. Hoffmann-La Roche
Curated by PDSP Ki Database
F. Hoffmann-La Roche
Curated by PDSP Ki Database
Affinity DataKi: 12nMAssay Description:Displacement by compound of [3H]-3-methoxy-5-(pyridin-2-ylethynyl)pyridine from rat cortical membranesMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
F. Hoffmann-La Roche
Curated by PDSP Ki Database
F. Hoffmann-La Roche
Curated by PDSP Ki Database
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
F. Hoffmann-La Roche
Curated by PDSP Ki Database
F. Hoffmann-La Roche
Curated by PDSP Ki Database
Affinity DataKi: 16nMAssay Description:Displacement of [3H]methoxy-PEPY from rat mGluR5 expressed in human HEK-293 cells by liquid scintillation countingMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
F. Hoffmann-La Roche
Curated by PDSP Ki Database
F. Hoffmann-La Roche
Curated by PDSP Ki Database
Affinity DataKi: 16nMAssay Description:Tested for displacement of [3H]3-methoxy-5-(pyridin-2-ylethynyl) pyridine from Metabotropic glutamate receptor 5 in rat cortical membraneMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
F. Hoffmann-La Roche
Curated by PDSP Ki Database
F. Hoffmann-La Roche
Curated by PDSP Ki Database
Affinity DataKi: 16nMAssay Description:Displacement of [3HMPEP from rat cloned mGluR5 expressed in HEK293T cells by by scintillation countingMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
F. Hoffmann-La Roche
Curated by PDSP Ki Database
F. Hoffmann-La Roche
Curated by PDSP Ki Database
Affinity DataKi: 16nMAssay Description:Displacement of [3H]-3-methoxy-5-(pyridin-2-ylethynyl)pyridine from mGlu5R in rat cortical membranes by liquid scintillation spectrometric analysisMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
F. Hoffmann-La Roche
Curated by PDSP Ki Database
F. Hoffmann-La Roche
Curated by PDSP Ki Database
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
F. Hoffmann-La Roche
Curated by PDSP Ki Database
F. Hoffmann-La Roche
Curated by PDSP Ki Database
Affinity DataKi: 33nMAssay Description:Displacement of [3H]MPEP from human cloned mGluR5 receptor expressed in CHO-T-Rex cells after 60 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
F. Hoffmann-La Roche
Curated by PDSP Ki Database
F. Hoffmann-La Roche
Curated by PDSP Ki Database
Affinity DataKi: 33nMAssay Description:Displacement of [3H]MPEP from human mGlu5 receptor expressed in CHO-TREx cell membranes after 60 mins by liquid scintillation spectrometric analysisMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Homo sapiens (Human))
F. Hoffmann-La Roche
Curated by PDSP Ki Database
F. Hoffmann-La Roche
Curated by PDSP Ki Database
Affinity DataKi: 33nMAssay Description:Displacement of [3H]MPEP from human mGlu5 receptor expressed in CHO-TREx cell membranes after 60 mins by liquid scintillation spectrometric analysisMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
F. Hoffmann-La Roche
Curated by PDSP Ki Database
F. Hoffmann-La Roche
Curated by PDSP Ki Database
Affinity DataKi: 39nMAssay Description:Displacement of [3H]MPEP from mGluR5 receptor in Sprague-Dawley rat forebrain membrane after 60 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
F. Hoffmann-La Roche
Curated by PDSP Ki Database
F. Hoffmann-La Roche
Curated by PDSP Ki Database
Affinity DataKi: 42nMAssay Description:Displacement of [3H]MPEP from mGluR5 in Sprague-Dawley rat brain membrane after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 500nMAssay Description:Competitive inhibition of CYP1A2 in human liver microsomes using phenacetin as substrate after 20 mins by LC-MS/MS analysisMore data for this Ligand-Target Pair
Affinity DataKi: 500nMAssay Description:Competitive inhibition of CYP1A2 in human liver microsomes using phenacetin as substrate after 20 mins by LC-MS/MS analysisMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]MPEP from rat mGlu1 receptor expressed in CHO-TREx cell membranes after 30 mins by liquid scintillation spectrometric analysisMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]MPEP from rat mGlu1 receptor expressed in CHO-TREx cell membranes after 30 mins by liquid scintillation spectrometric analysisMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]R214127 from rat cloned mGluR1 receptor expressed in CHO-T-Rex cells after 30 mins by liquid scintillation spectrometryMore data for this Ligand-Target Pair