Compile Data Set for Download or QSAR
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Found 3 of ki for monomerid = 50173176
TargetAdenosine receptor A2a(Rattus norvegicus (rat))
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50173176(8-Amino-2-furan-2-yl-[1,2,4]triazolo[1,5-a]pyrazin...)
Affinity DataKi:  1nMAssay Description:Binding affinity towards adenosine A2a receptor of rat brain homogenates using [3H]-ZM-241,385 compared to SCH-58261 (Ki=37 nM)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Leiden/Amsterdam Center For Drug Research

Curated by ChEMBL
LigandPNGBDBM50173176(8-Amino-2-furan-2-yl-[1,2,4]triazolo[1,5-a]pyrazin...)
Affinity DataKi:  1nMAssay Description:Binding affinity to human adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Biogen Idec

Curated by ChEMBL
LigandPNGBDBM50173176(8-Amino-2-furan-2-yl-[1,2,4]triazolo[1,5-a]pyrazin...)
Affinity DataKi:  320nMAssay Description:Binding affinity towards adenosine A1 receptor of rat cerebral cortex using [3H]-DPCPX compared to SCH-58261 (Ki=390 nM)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed