Compile Data Set for Download or QSAR
maximum 50k data
Found 4 of ki for monomerid = 50185331
TargetGamma-aminobutyric acid receptor subunit alpha-1/beta-3/gamma-2(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50185331(5-[4-fluoro-3-(3,5-difluoropyridin-2-yl)-phenyl]-3...)
Affinity DataKi:  1.5nMAssay Description:Displacement of [3H]Ro15-1788 from recombinant human GABA-Aalpha1 receptor plus beta3gamma2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-aminobutyric acid receptor subunit alpha-3/beta-3/gamma-2(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50185331(5-[4-fluoro-3-(3,5-difluoropyridin-2-yl)-phenyl]-3...)
Affinity DataKi:  8.5nMAssay Description:Displacement of [3H]Ro15-1788 from recombinant human GABA-Aalpha3 receptor plus beta3gamma2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGABA-A receptor; alpha-2/beta-3/gamma-2(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50185331(5-[4-fluoro-3-(3,5-difluoropyridin-2-yl)-phenyl]-3...)
Affinity DataKi:  10.9nMAssay Description:Displacement of [3H]Ro15-1788 from recombinant human GABA-Aalpha2 receptor plus beta3gamma2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGABA-A receptor; alpha-5/beta-3/gamma-2(Homo sapiens (Human))
Merck Sharp & Dohme Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50185331(5-[4-fluoro-3-(3,5-difluoropyridin-2-yl)-phenyl]-3...)
Affinity DataKi:  12.1nMAssay Description:Displacement of [3H]Ro15-1788 from recombinant human GABA-Aalpha5 receptor plus beta3gamma2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed