Compile Data Set for Download or QSAR
maximum 50k data
Found 3 of ki for monomerid = 50279280
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Università

Curated by ChEMBL
LigandPNGBDBM50279280(1-(4-Fluorophenyl)-3-(cytisin-12-yl)-1-propanone |...)
Affinity DataKi:  5.30nMAssay Description:Displacement of (+/-)-[3H]epibatidine from alpha4beta2 nicotinic acetylcholine receptor in rat brain cortex membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Università

Curated by ChEMBL
LigandPNGBDBM50279280(1-(4-Fluorophenyl)-3-(cytisin-12-yl)-1-propanone |...)
Affinity DataKi:  13nMAssay Description:Displacement of [3H]cytisine from alpha4beta2 nicotinic acetylcholine receptor in rat brain cortex membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Rattus norvegicus (Rat))
Università

Curated by ChEMBL
LigandPNGBDBM50279280(1-(4-Fluorophenyl)-3-(cytisin-12-yl)-1-propanone |...)
Affinity DataKi:  433nMAssay Description:Displacement of [125I]alpha-bungarotoxin from alpha7 nicotinic acetylcholine receptor in rat brain cortex membrane homogenatesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed