Compile Data Set for Download or QSAR
maximum 50k data
Found 7 of ki for monomerid = 50451054
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Dipartimento Di Farmacia Universit£

Curated by ChEMBL
LigandPNGBDBM50451054(CHEMBL4208744)
Affinity DataKi:  0.183nMAssay Description:Displacement of [3H]-8-OH-DPAT from serotonin 5-HT1A receptor in Sprague-Dawley rat brain cortex homogenates incubated for 30 mins by liquid scintill...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Dipartimento Di Farmacia Universit£

Curated by ChEMBL
LigandPNGBDBM50451054(CHEMBL4208744)
Affinity DataKi:  31nMAssay Description:Displacement of [3H]prazosin from adrenergic alpha1 receptor in rat cerebral cortexMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Rattus norvegicus (rat))
Dipartimento Di Farmacia Universit£

Curated by ChEMBL
LigandPNGBDBM50451054(CHEMBL4208744)
Affinity DataKi:  74nMAssay Description:Displacement of [3H]ketanserin from serotonin 5-HT2A receptor in Sprague-Dawley rat brain cortex homogenates incubated for 15 mins by liquid scintill...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
Dipartimento Di Farmacia Universit£

Curated by ChEMBL
LigandPNGBDBM50451054(CHEMBL4208744)
Affinity DataKi:  250nMAssay Description:Displacement of [3H]methyl-spiperone from human recombinant dopamine D2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Dipartimento Di Farmacia Universit£

Curated by ChEMBL
LigandPNGBDBM50451054(CHEMBL4208744)
Affinity DataKi:  610nMAssay Description:Displacement of [3H]SCH-23390 from human recombinant dopamine D1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50451054(CHEMBL4208744)
Affinity DataKi:  4.20E+3nMAssay Description:Displacement of [3H]RX 821002 from adrenergic alpha2 receptor in rat cerebral cortexMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
Dipartimento Di Farmacia Universit£

Curated by ChEMBL
LigandPNGBDBM50451054(CHEMBL4208744)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]mesulergine from serotonin 5-HT2C receptor in Sprague-Dawley rat brain cortex homogenates incubated for 15 mins by liquid scintil...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed