TargetD(4) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander-Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander-Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataKi: 0.25nMAssay Description:Displacement of [3H] Spiperone from human D4.4 receptor expressed in CHO cells by competitive radioligand binding assayMore data for this Ligand-Target Pair
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Friedrich-Alexander-Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander-Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataKi: 1.70nMAssay Description:Displacement of [3H] prazosin from alpha1A adrenergic receptor (unknown origin)More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 1A(Homo sapiens (Human))
Friedrich-Alexander-Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander-Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataKi: 17nMAssay Description:Displacement of [3H] WAY100635 from 5HT1A receptor (unknown origin)More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Friedrich-Alexander-Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander-Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataKi: 65nMAssay Description:Displacement of [3H] Ketanserin from 5HT2A receptor (unknown origin)More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander-Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander-Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataKi: 73nMAssay Description:Displacement of [3H] Spiperone from human D2S receptor expressed in CHO cells by competitive radioligand binding assayMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander-Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander-Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataKi: 77nMAssay Description:Displacement of [3H] Spiperone from human D2L receptor expressed in CHO cells by competitive radioligand binding assayMore data for this Ligand-Target Pair
TargetD(3) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander-Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander-Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataKi: 170nMAssay Description:Displacement of [3H] Spiperone from human D3 receptor expressed in CHO cells by competitive radioligand binding assayMore data for this Ligand-Target Pair
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander-Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander-Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataKi: 200nMAssay Description:Displacement of [3H] SCH23390 from D1 receptor (unknown origin)More data for this Ligand-Target Pair
TargetD(1B) dopamine receptor(Homo sapiens (Human))
Friedrich-Alexander-Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander-Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataKi: 340nMAssay Description:Displacement of [3H] SCH23390 from D5 receptor (unknown origin)More data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Friedrich-Alexander-Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander-Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataKi: 400nMAssay Description:Displacement of [3H] RX821002 from alpha2A adrenergic receptor (unknown origin)More data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Friedrich-Alexander-Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander-Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataKi: 1.80E+3nMAssay Description:Displacement of [3H] CGP12177 from beta2 adrenergic receptor (unknown origin)More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
Friedrich-Alexander-Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander-Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataKi: 2.00E+3nMAssay Description:Displacement of [3H] diprenorphine from mu opioid receptor (unknown origin)More data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Homo sapiens (Human))
Friedrich-Alexander-Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander-Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataKi: 3.90E+3nMAssay Description:Displacement of [3H] diprenorphine from kappa opioid receptor (unknown origin)More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Friedrich-Alexander-Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander-Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataKi: 1.00E+4nMAssay Description:Displacement of [3H] diprenorphine from delta opioid receptor (unknown origin)More data for this Ligand-Target Pair
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Friedrich-Alexander-Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander-Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataKi: 1.30E+4nMAssay Description:Displacement of [3H] CGP12177 from beta1 adrenergic receptor (unknown origin)More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Friedrich-Alexander-Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander-Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataKi: 1.40E+4nMAssay Description:Displacement of [3H] NMS from muscarinic M2 receptor (unknown origin)More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Friedrich-Alexander-Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander-Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataKi: 2.50E+4nMAssay Description:Displacement of [3H] NMS from muscarinic M3 receptor (unknown origin)More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Friedrich-Alexander-Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander-Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataKi: 2.50E+4nMAssay Description:Displacement of [3H] NMS from muscarinic M1 receptor (unknown origin)More data for this Ligand-Target Pair