Compile Data Set for Download or QSAR
maximum 50k data
Found 8 of ki for monomerid = 50525155
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
University Of South Australia

Curated by ChEMBL
LigandPNGBDBM50525155(CHEMBL4561424)
Affinity DataKi:  160nMAssay Description:Inhibition of recombinant full length N-terminal GST tagged human CDK5/p25 expressed in baculovirus infected sf9 cells using histone H1 as substrate ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
University Of South Australia

Curated by ChEMBL
LigandPNGBDBM50525155(CHEMBL4561424)
Affinity DataKi:  270nMAssay Description:Inhibition of recombinant full length N-terminal GST tagged human CDK2/CyclinA expressed in baculovirus infected sf9 cells using histone H1 as substr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
University Of South Australia

Curated by ChEMBL
LigandPNGBDBM50525155(CHEMBL4561424)
Affinity DataKi:  1.00E+3nMAssay Description:Inhibition of CDK2/Cyclin E (unknown origin) incubated for 30 to 120 mins in presence of ATP by ADP-Glo kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetCyclin-T1/Cyclin-dependent kinase 9(Homo sapiens (Human))
University Of South Australia

Curated by ChEMBL
LigandPNGBDBM50525155(CHEMBL4561424)
Affinity DataKi:  1.00E+3nMAssay Description:Inhibition of human recombinant full length N-terminal GST His6 fused CDK9 (M1 to F372 residues/ N-terminal His6 tagged Cyclin T1 (M1 to K726 residue...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
University Of South Australia

Curated by ChEMBL
LigandPNGBDBM50525155(CHEMBL4561424)
Affinity DataKi:  2.61E+3nMAssay Description:Inhibition of CDK1/CyclinB1 (unknown origin) using histone H1 (GGGPATPKKAKKL) as substrate incubated for 80 mins in presence of ATP by ADP-Glo kinase...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetCyclin-dependent kinase 6/G1/S-specific cyclin-D3(Homo sapiens (Human))
University Of South Australia

Curated by ChEMBL
LigandPNGBDBM50525155(CHEMBL4561424)
Affinity DataKi:  3.01E+3nMAssay Description:Inhibition of human recombinant N-terminal GST-tagged CDK6 (M1-A326 residues) and His6 tagged Cyclin D3 (M1-L292 residues) expressed in sf9 cells usi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetCDK-activating kinase assembly factor MAT1/Cyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
University Of South Australia

Curated by ChEMBL
LigandPNGBDBM50525155(CHEMBL4561424)
Affinity DataKi: >5.00E+3nMAssay Description:Inhibition of CDK7/cyclinH/MAT1 (unknown origin) using RBER-IRStide as substrate incubated for 120 mins in presence of ATP by ADP-Glo kinase assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
University Of South Australia

Curated by ChEMBL
LigandPNGBDBM50525155(CHEMBL4561424)
Affinity DataKi: >5.00E+3nMAssay Description:Inhibition of human recombinant N-terminal GST-tagged CDK4 (S4-E303 residues)/Cyclin D1 (Q4-I295 residues) expressed in sf9 cells using RB-CTF as sub...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed