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Found 6 Enz. Inhib. hit(s) with Target = '5-hydroxytryptamine receptor 4' and Ligand = 'BDBM85027'
Target5-hydroxytryptamine receptor 4(RAT)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM85027(1-(7-Chloro-8-amino-1,4-benzodioxane-5-yl)-3-[1-[3...)
Affinity DataKi:  0.000400nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(RAT)
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM85027(1-(7-Chloro-8-amino-1,4-benzodioxane-5-yl)-3-[1-[3...)
Affinity DataKi:  0.000480nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM85027(1-(7-Chloro-8-amino-1,4-benzodioxane-5-yl)-3-[1-[3...)
Affinity DataKi:  0.000580nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Cnrs Upr 9023

Curated by PDSP Ki Database
LigandPNGBDBM85027(1-(7-Chloro-8-amino-1,4-benzodioxane-5-yl)-3-[1-[3...)
Affinity DataKi:  0.000630nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Roche Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM85027(1-(7-Chloro-8-amino-1,4-benzodioxane-5-yl)-3-[1-[3...)
Affinity DataKi:  0.100nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 4(GUINEA PIG)
Roche Bioscience

Curated by PDSP Ki Database
LigandPNGBDBM85027(1-(7-Chloro-8-amino-1,4-benzodioxane-5-yl)-3-[1-[3...)
Affinity DataKi:  0.100nMAssay Description:Compound was evaluated for binding affinity against 5-hydroxytryptamine 4 receptor using radioligand binding assay using [3H]GR as radioligandMore data for this Ligand-Target Pair
In DepthDetails