Compile Data Set for Download or QSAR
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Found 5 Enz. Inhib. hit(s) with Target = 'Peroxisome proliferator-activated receptor alpha' and Ligand = 'BDBM50171897'
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50171897((2S)-2-(4-chlorophenoxy)-3-phenylpropanoic acid | ...)
Affinity DataEC50:  3.90E+3nMAssay Description:Effective concentration against human PPARalpha expressed in HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Mus musculus)
Università

Curated by ChEMBL
LigandPNGBDBM50171897((2S)-2-(4-chlorophenoxy)-3-phenylpropanoic acid | ...)
Affinity DataEC50:  1.30nMAssay Description:Effective concentration against murine PPARalpha in transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50171897((2S)-2-(4-chlorophenoxy)-3-phenylpropanoic acid | ...)
Affinity DataEC50:  3.89E+3nMAssay Description:Agonist activity at GAL4-fused PPARalpha (unknown origin) expressed in human HepG2 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50171897((2S)-2-(4-chlorophenoxy)-3-phenylpropanoic acid | ...)
Affinity DataEC50:  4.90E+3nMAssay Description:Agonist activity at GAL4-tagged human PPARalpha ligand binding domain expressed in HepG2 cells assessed as transactivation after 20 hrs by beta-galac...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50171897((2S)-2-(4-chlorophenoxy)-3-phenylpropanoic acid | ...)
Affinity DataEC50:  1.45E+4nMAssay Description:Agonist activity at human PPARalpha ligand binding domain expressed in human HepG2 cells cotransfected with Gal4 by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed