Found 12 Enz. Inhib. hit(s) with Target = 'Retinoic acid receptor RXR-alpha' and Ligand = 'BDBM50032671'
Affinity DataKi: 3nMAssay Description:Binding affinity against Retinoic acid receptor RXR-alpha by [3H]-9-cis-RA displacement.More data for this Ligand-Target Pair
Affinity DataKi: 13nMAssay Description:In vitro agonistic activity against PPAR gamma along with 100 nM BRL49653More data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Binding affinity against Retinoic acid receptor RXR-alpha was determined in vitro by using [3H]-9-cis-RA as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:In vitro inhibition of 5-(125I)A-85380 binding to nicotinic acetylcholine receptor (nAChR) of rat brainMore data for this Ligand-Target Pair
Affinity DataIC50: 5nMAssay Description:Invitro evaluation against RXR-alpha in CV-1 cells by cotransfection assay was determinedMore data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Antagonist activity for Retinoic X receptor alpha in CV1 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 40nMAssay Description:Activation of human RXRalpha activity expressed in COS1 cells after 12 hrs by RXRE-luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 11nMAssay Description:Inhibition of Retinoic acid receptor RXR-alpha agonist activity in vitroMore data for this Ligand-Target Pair
Affinity DataKd: 3nMAssay Description:Ability to bind directly to Retinoic acid receptor RXR-alpha was evaluated in a competitive binding assay.More data for this Ligand-Target Pair
Affinity DataEC50: 4nMAssay Description:Ability to activate gene expression at Retinoic acid receptor RXR-alpha was evaluated in a cotransfection assay.More data for this Ligand-Target Pair
Affinity DataEC50: 17nMAssay Description:In vitro agonistic activity against RXR alpha in CV-1 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 11nMAssay Description:In vitro transcriptional activation in CV-1 cells expressing RXR-alphaMore data for this Ligand-Target Pair