Compile Data Set for Download or QSAR
Report error Found 4 Enz. Inhib. hit(s) with Target = 'Tyrosine-protein kinase BTK' and Ligand = 'BDBM143185'
TargetTyrosine-protein kinase BTK(Human)
Principia Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 143185BDBM143185(US9266895, 10 | US8940744, 10 | US9994576, 10 | US...)
Affinity DataIC50: 2.10nMAssay Description:A Caliper-based kinase assay (Caliper Life Sciences, Hopkinton, Mass.) was used to measure inhibition of Btk kinase activity of a compound of the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/5/2020
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Principia Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 143185BDBM143185(US9266895, 10 | US8940744, 10 | US9994576, 10 | US...)
Affinity DataIC50: 2.10nMT: 2°CAssay Description:A Caliper-based kinase assay (Caliper Life Sciences, Hopkinton, Mass.) was used to measure inhibition of Btk kinase activity of a compound of the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/17/2017
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Principia Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 143185BDBM143185(US9266895, 10 | US8940744, 10 | US9994576, 10 | US...)
Affinity DataIC50: 2.10nMT: 2°CAssay Description:A Caliper-based kinase assay (Caliper Life Sciences, Hopkinton, Mass.) was used to measure inhibition of Btk kinase activity of a compound of the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2015
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Principia Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 143185BDBM143185(US9266895, 10 | US8940744, 10 | US9994576, 10 | US...)
Affinity DataIC50: 2.10nMAssay Description:A Caliper-based kinase assay (Caliper Life Sciences, Hopkinton, Mass.) was used to measure inhibition of Btk kinase activity of a compound of the pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2021
Entry Details
US Patent