Filter my 2727 hits
Targets 352▿
Aurora kinase B 66
Serine/threonine-protein kinase B-raf 63
Receptor-type tyrosine-protein kinase FLT3 42
Aurora kinase A 38
Tyrosine-protein kinase JAK1 15
Ribosomal protein S6 kinase alpha-2 14
Ribosomal protein S6 kinase alpha-1 14
Ephrin type-A receptor 6 14
Non-receptor tyrosine-protein kinase TYK2 14
Mitogen-activated protein kinase 14 14
Myosin light chain kinase, smooth muscle 14
Serine/threonine-protein kinase TAO1 14
Ribosomal protein S6 kinase alpha-6 14
Calcium/calmodulin-dependent protein kinase type II subunit gamma 14
Ribosomal protein S6 kinase alpha-4 14
Ribosomal protein S6 kinase alpha-5 14
Mast/stem cell growth factor receptor Kit 9
Proto-oncogene tyrosine-protein kinase receptor Ret 9
Platelet-derived growth factor receptor beta 9
Macrophage colony-stimulating factor 1 receptor 9
Vascular endothelial growth factor receptor 2 9
Aurora kinase C 9
Mitogen-activated protein kinase 1 8
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform 8
Serine/threonine-protein kinase PLK1 8
Tyrosine-protein kinase Lck 8
Mitogen-activated protein kinase 3 8
Ephrin type-A receptor 2 8
Tyrosine-protein kinase ABL1 8
RAF proto-oncogene serine/threonine-protein kinase 8
Platelet-derived growth factor receptor alpha 8
Epidermal growth factor receptor 8
Dual specificity mitogen-activated protein kinase kinase 2 8
Tyrosine-protein kinase JAK3 8
Tyrosine-protein kinase JAK2 8
Dual specificity mitogen-activated protein kinase kinase 1 8
ALK tyrosine kinase receptor 8
Hepatocyte growth factor receptor 8
Epithelial discoidin domain-containing receptor 1 8
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit beta isoform 8
Insulin receptor 8
Vascular endothelial growth factor receptor 3 8
Vascular endothelial growth factor receptor 1 8
Tyrosine-protein kinase Tec 7
BMP-2-inducible protein kinase 7
Rhodopsin kinase GRK1 7
Cyclin-dependent kinase 11B 7
Cyclin-dependent kinase 11A 7
Uncharacterized serine/threonine-protein kinase SBK3 7
LIM domain kinase 1 7
LIM domain kinase 2 7
NUAK family SNF1-like kinase 2 7
Glycogen synthase kinase-3 beta 7
Calcium/calmodulin-dependent protein kinase type 1 7
NUAK family SNF1-like kinase 1 7
AP2-associated protein kinase 1 7
Calcium/calmodulin-dependent protein kinase type II subunit beta 7
Phosphorylase b kinase gamma catalytic chain, skeletal muscle/heart isoform 7
Serine/threonine-protein kinase PAK 1 7
Protein kinase C theta type 7
Serine/threonine-protein kinase PAK 2 7
Serine/threonine-protein kinase PAK 3 7
Serine/threonine-protein kinase PAK 4 7
Phosphatidylinositol 5-phosphate 4-kinase type-2 beta 7
Serine/threonine-protein kinase tousled-like 2 7
Dual specificity mitogen-activated protein kinase kinase 3 7
Serine/threonine-protein kinase PAK 5 7
Serine/threonine-protein kinase PAK 6 7
Serine/threonine-protein kinase tousled-like 1 7
Protein delta homolog 1 7
Dual specificity mitogen-activated protein kinase kinase 6 7
Dual specificity mitogen-activated protein kinase kinase 4 7
Tyrosine-protein kinase ZAP-70 7
Casein kinase I isoform gamma-3 7
Casein kinase I isoform gamma-2 7
Casein kinase I isoform epsilon 7
Casein kinase I isoform gamma-1 7
Ephrin type-A receptor 1 7
Ephrin type-A receptor 3 7
Ephrin type-A receptor 5 7
Tyrosine-protein kinase BTK 7
Ephrin type-A receptor 4 7
Tyrosine-protein kinase receptor UFO 7
Insulin-like growth factor 1 receptor 7
Activin receptor type-1 7
Myosin light chain kinase 2, skeletal/cardiac muscle 7
Tyrosine-protein kinase Srms 7
Wee1-like protein kinase 7
U4/U6 small nuclear ribonucleoprotein Prp4 7
Serine/threonine-protein kinase/endoribonuclease IRE1 7
Serine/threonine-protein kinase MAK 7
Phosphatidylinositol 3-kinase C2 domain-containing subunit gamma 7
Ankyrin repeat and protein kinase domain-containing protein 1 7
Tyrosine-protein kinase Lyn 7
Focal adhesion kinase 1 7
Cyclin-dependent kinase 2 7
Tyrosine-protein kinase TXK 7
Rhodopsin kinase GRK7 7
Ephrin type-A receptor 8 7
Phosphatidylinositol 4-kinase beta 7
Death-associated protein kinase 2 7
Death-associated protein kinase 1 7
Serine/threonine-protein kinase D2 7
Serine/threonine-protein kinase D3 7
TGF-beta receptor type-2 7
Serine/threonine-protein kinase D1 7
Dual specificity tyrosine-phosphorylation-regulated kinase 1B 7
Dual specificity tyrosine-phosphorylation-regulated kinase 1A 7
Death-associated protein kinase 3 7
Cyclin-dependent kinase 9 7
Serine/threonine-protein kinase pim-3 7
Cyclin-dependent kinase 8 7
Cyclin-dependent kinase 7 7
Serine/threonine-protein kinase pim-1 7
Cyclin-dependent kinase 5 7
Serine/threonine-protein kinase pim-2 7
Serine/threonine-protein kinase 38 7
Serine/threonine-protein kinase 35 7
Cyclin-dependent kinase 3 7
Serine/threonine-protein kinase 36 7
Cyclin-dependent kinase 16 7
Testis-specific serine/threonine-protein kinase 1 7
Protein kinase C epsilon type 7
Cyclin-dependent kinase 17 7
Bone morphogenetic protein receptor type-2 7
Cyclin-dependent kinase 19 7
Protein-tyrosine kinase 6 7
Casein kinase II subunit alpha 7
Cyclin-dependent kinase 14 7
Cyclin-dependent kinase 15 7
Leukocyte tyrosine kinase receptor 7
Cytoplasmic tyrosine-protein kinase BMX 7
Tyrosine-protein kinase ABL2 7
Atypical kinase COQ8B, mitochondrial 7
Microtubule-associated serine/threonine-protein kinase 1 7
Calcium/calmodulin-dependent protein kinase type II subunit alpha 7
cGMP-dependent protein kinase 2 7
Rho-associated protein kinase 2 7
cGMP-dependent protein kinase 1 7
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit gamma isoform 7
Rho-associated protein kinase 1 7
Serine/threonine-protein kinase ULK1 7
Serine/threonine-protein kinase SIK2 7
Tyrosine-protein kinase Fes/Fps 7
Serine/threonine-protein kinase SIK1 7
Serine/threonine-protein kinase ULK2 7
Serine/threonine-protein kinase ULK3 7
3-phosphoinositide-dependent protein kinase 1 7
Serine/threonine-protein kinase 3 7
Discoidin domain-containing receptor 2 7
Mitogen-activated protein kinase 4 7
Serine/threonine-protein kinase 4 7
SRSF protein kinase 3 7
Mitogen-activated protein kinase 9 7
SRSF protein kinase 2 7
Mitogen-activated protein kinase 6 7
Mitogen-activated protein kinase 7 7
Calcium/calmodulin-dependent protein kinase type IV 7
Mitogen-activated protein kinase 8 7
Tyrosine-protein kinase SYK 7
Serine/threonine-protein kinase TBK1 7
Serine/threonine-protein kinase RIO1 7
Serine/threonine-protein kinase LATS1 7
Serine/threonine-protein kinase RIO3 7
Serine/threonine-protein kinase 32B 7
Serine/threonine-protein kinase RIO2 7
Serine/threonine-protein kinase 32C 7
Tyrosine-protein kinase HCK 7
Serine/threonine-protein kinase PLK2 7
Insulin receptor-related protein 7
Inhibitor of nuclear factor kappa-B kinase subunit beta 7
Serine/threonine-protein kinase NIM1 7
Serine/threonine-protein kinase PLK3 7
Serine/threonine-protein kinase PLK4 7
Tyrosine-protein kinase receptor TYRO3 7
Wee1-like protein kinase 2 7
Serine/threonine-protein kinase BRSK1 7
Serine/threonine-protein kinase LATS2 7
Citron Rho-interacting kinase 7
Serine/threonine-protein kinase BRSK2 7
Serine/threonine-protein kinase Chk2 7
Serine/threonine-protein kinase Chk1 7
cAMP-dependent protein kinase catalytic subunit PRKX 7
SRSF protein kinase 1 7
Tyrosine-protein kinase Yes 7
Serine/threonine-protein kinase MRCK beta 7
Serine/threonine-protein kinase MRCK gamma 7
Casein kinase II subunit alpha' 7
Dual specificity tyrosine-phosphorylation-regulated kinase 2 7
Serine/threonine-protein kinase STK11 7
Cyclin-G-associated kinase 7
Receptor tyrosine-protein kinase erbB-4 7
Receptor tyrosine-protein kinase erbB-2 7
Tyrosine-protein kinase FRK 7
Receptor tyrosine-protein kinase erbB-3 7
Phosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit delta isoform 7
Serine/threonine-protein kinase Nek9 7
Serine/threonine-protein kinase Nek7 7
Glycogen synthase kinase-3 alpha 7
Serine/threonine-protein kinase Nek6 7
Serine/threonine-protein kinase Nek5 7
Serine/threonine-protein kinase Nek2 7
Serine/threonine-protein kinase receptor R3 7
Serine/threonine-protein kinase Nek1 7
Macrophage-stimulating protein receptor 7
Cyclin-dependent kinase-like 3 7
Serine/threonine-protein kinase SIK3 [59-1321] 7
Cyclin-dependent kinase-like 2 7
MAP/microtubule affinity-regulating kinase 3 7
Homeodomain-interacting protein kinase 4 7
Homeodomain-interacting protein kinase 3 7
MAP kinase-interacting serine/threonine-protein kinase 2 7
MAP kinase-interacting serine/threonine-protein kinase 1 7
Cyclin-dependent kinase-like 5 7
Membrane-associated tyrosine- and threonine-specific cdc2-inhibitory kinase 7
Serine/threonine-protein kinase 10 7
MAP/microtubule affinity-regulating kinase 4 7
Serine/threonine-protein kinase 38-like 7
Dual specificity protein kinase TTK 7
Myosin-IIIb 7
Myosin-IIIa 7
Tyrosine-protein kinase ITK/TSK 7
Myotonin-protein kinase 7
Protein kinase C eta type 7
Bone morphogenetic protein receptor type-1B 7
Bone morphogenetic protein receptor type-1A 7
Tyrosine-protein kinase Blk 7
Receptor-interacting serine/threonine-protein kinase 1 7
Serine/threonine-protein kinase 16 7
Receptor-interacting serine/threonine-protein kinase 2 7
Non-receptor tyrosine-protein kinase TNK1 7
Inhibitor of nuclear factor kappa-B kinase subunit epsilon 7
Serine/threonine-protein kinase NLK 7
Homeodomain-interacting protein kinase 2 7
Homeodomain-interacting protein kinase 1 7
Receptor-interacting serine/threonine-protein kinase 4 7
Ribosomal protein S6 kinase beta-1 7
Serine/threonine-protein kinase OSR1 7
Casein kinase I isoform delta 7
Cyclin-dependent kinase 18 [3-474] 7
Serine/threonine-protein kinase 26 7
Serine/threonine-protein kinase 24 7
Serine/threonine-protein kinase 25 7
Dual specificity testis-specific protein kinase 1 7
Ephrin type-B receptor 3 7
Serine/threonine-protein kinase 33 7
Ephrin type-B receptor 4 7
Ephrin type-B receptor 1 7
Ephrin type-B receptor 2 7
MAP kinase-activated protein kinase 2 7
Ephrin type-B receptor 6 7
MAP kinase-activated protein kinase 5 7
STE20/SPS1-related proline-alanine-rich protein kinase 7
Muscle, skeletal receptor tyrosine-protein kinase 7
Tyrosine-protein kinase Fer 7
Tyrosine-protein kinase receptor Tie-1 7
5'-AMP-activated protein kinase catalytic subunit alpha-2 7
Calcium/calmodulin-dependent protein kinase type II subunit delta 7
Proto-oncogene tyrosine-protein kinase ROS 7
Serine/threonine-protein kinase DCLK1 7
Calcium/calmodulin-dependent protein kinase kinase 1 7
Serine/threonine-protein kinase DCLK2 7
Serine/threonine-protein kinase TAO3 7
Calcium/calmodulin-dependent protein kinase kinase 2 7
Serine/threonine-protein kinase DCLK3 7
Serine/threonine-protein kinase TNNI3K 7
Interferon-induced, double-stranded RNA-activated protein kinase 7
Angiopoietin-1 receptor 7
Mitogen-activated protein kinase kinase kinase kinase 2 7
Mitogen-activated protein kinase kinase kinase kinase 3 7
Mitogen-activated protein kinase kinase kinase kinase 1 7
Serine/threonine-protein kinase MRCK alpha 7
Mitogen-activated protein kinase kinase kinase kinase 4 7
Mitogen-activated protein kinase kinase kinase kinase 5 7
Mitogen-activated protein kinase 15 7
5'-AMP-activated protein kinase catalytic subunit alpha-1 7
Activin receptor type-1B 7
Myosin light chain kinase family member 4 7
Mitogen-activated protein kinase kinase kinase 9 7
Mitogen-activated protein kinase kinase kinase 6 7
RAC-gamma serine/threonine-protein kinase 7
Mitogen-activated protein kinase kinase kinase 5 7
Interleukin-1 receptor-associated kinase 1 7
Mitogen-activated protein kinase kinase kinase 7 7
Interleukin-1 receptor-associated kinase 3 7
Mitogen-activated protein kinase kinase kinase 2 7
Mitogen-activated protein kinase kinase kinase 1 7
Mitogen-activated protein kinase kinase kinase 4 7
Mitogen-activated protein kinase kinase kinase 3 7
Serine/threonine-protein kinase ICK 7
RAC-alpha serine/threonine-protein kinase 7
Megakaryocyte-associated tyrosine-protein kinase 7
Proto-oncogene tyrosine-protein kinase Src 7
Activin receptor type-2B 7
Activin receptor type-2A 7
BDNF/NT-3 growth factors receptor 7
Serine/threonine-protein kinase 17A 7
Serine/threonine-protein kinase 17B 7
Mitogen-activated protein kinase kinase kinase 19 7
Dual specificity protein kinase CLK1 7
Protein kinase C delta type 7
Mitogen-activated protein kinase kinase kinase 15 7
NT-3 growth factor receptor 7
G protein-coupled receptor kinase 4 7
Dual specificity protein kinase CLK4 7
Dual specificity protein kinase CLK3 7
Dual specificity protein kinase CLK2 7
High affinity nerve growth factor receptor 7
Protein-tyrosine kinase 2-beta 7
Tyrosine-protein kinase Mer 7
Poly [ADP-ribose] polymerase tankyrase-2 7
Serine/threonine-protein kinase N2 7
cAMP-dependent protein kinase catalytic subunit beta 7
Serine/threonine-protein kinase N1 7
Ribosomal protein S6 kinase alpha-3 7
Phosphorylase b kinase gamma catalytic chain, liver/testis isoform 7
Calcium/calmodulin-dependent protein kinase type 1D 7
STE20-like serine/threonine-protein kinase 7
Hormonally up-regulated neu tumor-associated kinase 7
Fibroblast growth factor receptor 4 7
Tyrosine-protein kinase Fgr 7
Phosphatidylinositol 4-phosphate 3-kinase C2 domain-containing subunit beta 7
Mitogen-activated protein kinase kinase kinase 20 7
Fibroblast growth factor receptor 1 7
Fibroblast growth factor receptor 2 7
Atypical kinase COQ8A, mitochondrial 7
Fibroblast growth factor receptor 3 7
Mitogen-activated protein kinase 13 7
Inhibitor of nuclear factor kappa-B kinase subunit alpha 7
Mitogen-activated protein kinase 12 7
Mitogen-activated protein kinase 11 7
Phosphatidylinositol 4-phosphate 5-kinase type-1 alpha 7
RAC-beta serine/threonine-protein kinase 7
Mitogen-activated protein kinase 10 7
Casein kinase I isoform alpha 7
Misshapen-like kinase 1 7
Tyrosine-protein kinase Fyn 7
Tyrosine-protein kinase CSK 7
Protein kinase C alpha type 7
Maternal embryonic leucine zipper kinase 7
Serine/threonine-protein kinase MARK1 7
Serine/threonine-protein kinase MARK2 7
TRAF2 and NCK-interacting protein kinase 7
Mitogen-activated protein kinase kinase kinase 13 7
Mitogen-activated protein kinase kinase kinase 10 7
Mitogen-activated protein kinase kinase kinase 11 7
Cytochrome P450 1A2 1
IGF-like family receptor 1 1
Cytochrome P450 2C9 1
Cytochrome P450 2C19 1
Cytochrome P450 2D6 1
Cytochrome P450 3A4 1
...
Publications 5▿
Blood 114: 2984 -92 (2009) 2521 J Med Chem 55: 3250 -60 (2012) 90 Bioorg Med Chem Lett 21: 5342 -6 (2011) 55 J Med Chem 55: 1082 -105 (2012) 32 J Med Chem 52: 7808 -16 (2009) 29
Institutions 1▿
Affinity: 0.075 to 7.5E+5 nM▿
Xtal structures: 4
Docked structures: 5
Catalog Cmpds: 10