TargetMas-related G-protein coupled receptor member X2(Homo sapiens (Human))
University of North Carolina
University of North Carolina
Affinity DataEC50: 1.10E+3nMpH: 7.4 T: 2°CAssay Description:MRGPRX2 stable cells were maintained in DMEM containing 10% FBS, 100 μg/ml hygromycin B, and 15 μg/ml blasticidin. For the calcium mobiliza...More data for this Ligand-Target Pair
TargetGrowth hormone secretagogue receptor type 1(Homo sapiens (Human))
Univ Montpellier
Curated by ChEMBL
Univ Montpellier
Curated by ChEMBL
Affinity DataEC50: 66nMAssay Description:Inverse agonist activity at SNAP-tagged human GHSR expressed in HEK293 cells assessed as inhibition of ghrelin-induced IP1 response measured after 30...More data for this Ligand-Target Pair
Affinity DataEC50: 1nMAssay Description:Agonist activity at tachykinin receptor 2 in the rat colon muscularis mucosaeMore data for this Ligand-Target Pair
Affinity DataEC50: 1nMAssay Description:Agonistic activity at tachykinin receptor 1 receptor in guinea pig ileum longitudinal smooth muscleMore data for this Ligand-Target Pair
Affinity DataEC50: 167nMAssay Description:Agonist activity at tachykinin receptor 2 in the rat colon muscularis mucosaeMore data for this Ligand-Target Pair
Affinity DataEC50: 4.90nMAssay Description:Agonistic activity at tachykinin receptor 1 receptor in guinea pig ileum longitudinal smooth muscleMore data for this Ligand-Target Pair
Affinity DataEC50: 5.60nMAssay Description:In vitro agonistic activity against tachykinin receptor 1 of guinea pig ileum longitudinal smooth muscle.More data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Marshall University School Of Medicine And Huntington Va Medical Center
Curated by ChEMBL
Marshall University School Of Medicine And Huntington Va Medical Center
Curated by ChEMBL
Affinity DataEC50: 1nMAssay Description:Agonist activity at bfSPR to produce increase in intracellular [Ca2+]More data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Marshall University School Of Medicine And Huntington Va Medical Center
Curated by ChEMBL
Marshall University School Of Medicine And Huntington Va Medical Center
Curated by ChEMBL
Affinity DataEC50: 0.600nMAssay Description:SP-induced [Ca2+] mobilization in CHO cells expressing human Tachykinin receptor 1More data for this Ligand-Target Pair
Affinity DataEC50: 167nMAssay Description:In vitro agonistic activity against tachykinin receptor 2 of rat colon muscularis mucosae.More data for this Ligand-Target Pair
Affinity DataEC50: 7.50E+3nMAssay Description:In vitro agonistic activity against tachykinin receptor 3 of everted rat protal vein.More data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Marshall University School Of Medicine And Huntington Va Medical Center
Curated by ChEMBL
Marshall University School Of Medicine And Huntington Va Medical Center
Curated by ChEMBL
Affinity DataEC50: 0.600nMAssay Description:Agonist activity at wild type human NK1 receptor expressed in HEK293 cells assessed as increase in [3H]IP accumulation after 20 minsMore data for this Ligand-Target Pair
TargetSubstance-P receptor(Homo sapiens (Human))
Marshall University School Of Medicine And Huntington Va Medical Center
Curated by ChEMBL
Marshall University School Of Medicine And Huntington Va Medical Center
Curated by ChEMBL
Affinity DataEC50: 0.0575nMAssay Description:Antagonist activity at human recombinant NK1 receptor expressed in CHO cells assessed as inhibition of NPS-induced intracellular calcium mobilizationMore data for this Ligand-Target Pair
Affinity DataEC50: 793nMAssay Description:Compound was evaluated for concentration-dependent and oscillatory increase in [Ca2+], caused by activation of hNK3 receptors in CHO cellsMore data for this Ligand-Target Pair
TargetMas-related G-protein coupled receptor member X2(Homo sapiens (Human))
University of North Carolina
University of North Carolina
Affinity DataEC50: 5.10E+3nMpH: 7.4 T: 2°CAssay Description:HTLA cells (HEK-T cells stably expressing a β-arrestin2-TEV fusion protein and a tTa-dependent luciferase reporter) were maintained in DMEM (Cor...More data for this Ligand-Target Pair