Affinity DataKi: 1nMAssay Description:Binding affinity to Homo sapiens (human) alpha1A adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Binding affinity to Homo sapiens (human) alpha1A adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Binding affinity determined by displacement of [3H]prazosin from alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:Binding affinity determined by displacement of [3H]prazosin from alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.87nMAssay Description:Binding affinity was determined for the alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 20.9nMAssay Description:Binding affinity determined by displacement of [3H]prazosin from alpha-1A adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 20.9nMAssay Description:Binding affinity to Homo sapiens (human) alpha1A adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
New York University Medical Center
Curated by ChEMBL
New York University Medical Center
Curated by ChEMBL
Affinity DataKi: 151nMAssay Description:Binding affinity determined by displacement of [3H]rauwolscine from alpha-2A adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
New York University Medical Center
Curated by ChEMBL
New York University Medical Center
Curated by ChEMBL
Affinity DataKi: 151nMAssay Description:Binding affinity determined by displacement of [3H]rauwolscine from alpha-2A adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
New York University Medical Center
Curated by ChEMBL
New York University Medical Center
Curated by ChEMBL
Affinity DataKi: 165nMAssay Description:Binding affinity assayed by displacement of [3H]rauwolscine from human alpha-2C adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
New York University Medical Center
Curated by ChEMBL
New York University Medical Center
Curated by ChEMBL
Affinity DataKi: 165nMAssay Description:Binding affinity assayed by displacement of [3H]rauwolscine from human alpha-2C adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-2C adrenergic receptor(Homo sapiens (Human))
New York University Medical Center
Curated by ChEMBL
New York University Medical Center
Curated by ChEMBL
Affinity DataKi: 166nMAssay Description:Binding affinity assayed by displacement of [3H]rauwolscine from human alpha-2C adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
New York University Medical Center
Curated by ChEMBL
New York University Medical Center
Curated by ChEMBL
Affinity DataKi: 223nMAssay Description:Binding affinity determined by displacement of [3H]prazosin from alpha-1D adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
New York University Medical Center
Curated by ChEMBL
New York University Medical Center
Curated by ChEMBL
Affinity DataKi: 224nMAssay Description:Binding affinity determined by displacement of [3H]prazosin from alpha-1D adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
New York University Medical Center
Curated by ChEMBL
New York University Medical Center
Curated by ChEMBL
Affinity DataKi: 281nMAssay Description:Binding affinity determined by displacement of [3H]rauwolscine from alpha-2B adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
New York University Medical Center
Curated by ChEMBL
New York University Medical Center
Curated by ChEMBL
Affinity DataKi: 281nMAssay Description:Binding affinity determined by displacement of [3H]rauwolscine from alpha-2B adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-2B adrenergic receptor(Homo sapiens (Human))
New York University Medical Center
Curated by ChEMBL
New York University Medical Center
Curated by ChEMBL
Affinity DataKi: 282nMAssay Description:Binding affinity determined by displacement of [3H]rauwolscine from alpha-2B adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
New York University Medical Center
Curated by ChEMBL
New York University Medical Center
Curated by ChEMBL
Affinity DataKi: 301nMAssay Description:Binding affinity determined by displacement of [3H]rauwolscine from alpha-2A adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 330nMAssay Description:Binding affinity was determined for the alpha-1B adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 331nMAssay Description:Binding affinity determined by displacement of [3H]prazosin from alpha-1B adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 363nMAssay Description:Binding affinity determined by displacement of [3H]prazosin from alpha-1B adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 363nMAssay Description:Binding affinity determined by displacement of [3H]prazosin from alpha-1B adrenergic receptorMore data for this Ligand-Target Pair
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
New York University Medical Center
Curated by ChEMBL
New York University Medical Center
Curated by ChEMBL
Affinity DataKi: 398nMAssay Description:Binding affinity determined by displacement of [3H]prazosin from alpha-1D adrenergic receptorMore data for this Ligand-Target Pair
Affinity DataKi: 600nMAssay Description:Binding affinity was determined for the alpha-1D adrenergic receptorMore data for this Ligand-Target Pair
TargetVoltage-dependent L-type calcium channel subunit alpha-1S(Rattus norvegicus)
New York University Medical Center
Curated by ChEMBL
New York University Medical Center
Curated by ChEMBL
Affinity DataKi: <1.00E+3nMAssay Description:Binding affinity at the L-type [Ca2+] channel from rat brain homogenate by [3H]nitrendipine displacement.More data for this Ligand-Target Pair